SCHEMBL11111670

SCHEMBL11111670

COc1ccc2c(c1)C(=CC(=O)O)c1ccccc1C=C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 3/20 0.40
AR P10275 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC2 Q92769 1/20 0.39
NTSR1 P30989 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
GPR3 P46089 1/20 0.38
MAPK1 P28482 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 1/20 0.38
PGR P06401 1/20 0.38
CYP2D6 P10635 1/20 0.38
HPGD P15428 1/20 0.38
SLC6A2 P23975 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11111667 1.00 HDAC8 (0.40) HDAC8ARHDAC4HDAC2NTSR1
SCHEMBL11117862 0.92 GPR3 (0.41) HDAC8ARNTSR1GPR3MAPK1
SCHEMBL11117865 0.92 GPR3 (0.41) HDAC8ARNTSR1GPR3MAPK1
SCHEMBL29454416 0.82 MEN1 (0.42) ALDH1A1CYP1A2LMNACYP2D6HPGD
SCHEMBL677773 0.82 MEN1 (0.42) ALDH1A1CYP1A2LMNACYP2D6HPGD
SCHEMBL1233660 0.79 MEN1 (0.49) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL11114767 0.78 TRPA1 (0.46) GPR3MAPTKDM4E
SCHEMBL11118131 0.78 S100A4 (0.38) ARALDH1A1HTT
SCHEMBL11115877 0.78 S100A4 (0.38) ARALDH1A1HTT
SCHEMBL11115874 0.78 S100A4 (0.38) ARALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0115690-A1 Dibenzocycloheptenylidenes AMERICAN HOME PRODUCTS CORPORATION (US) 1984-08-15 EP claimed
EP-0115690-A1 Dibenzocycloheptenylidenes AMERICAN HOME PRODUCTS CORPORATION (US) 1984-08-15 EP disclosed