SCHEMBL11114850

SCHEMBL11114850

CCC(C(=O)O)c1ccc(OCc2ccsc2C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.47
AKR1C2 P52895 5/20 0.47
AKR1C1 Q04828 1/20 0.47
PTGS1 P23219 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 2/20 0.40
FFAR1 O14842 2/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10984633 0.81 ALDH1A1 (0.39) ALDH1A1FFAR1NPC1RAB9ARXRA
SCHEMBL11115339 0.81 NPC1 (0.43) POLBALDH1A1FFAR1NPC1RAB9A
SCHEMBL11114869 0.78 ALDH1A1 (0.42) POLBALDH1A1FFAR1NPC1RAB9A
SCHEMBL8936259 0.78 SLC6A1 (0.51) FFAR1NPC1RAB9AMEN1KMT2A
SCHEMBL10988964 0.77 FFAR1 (0.40) POLBTDP1ALDH1A1FFAR1NPC1
SCHEMBL5757559 0.76 PTGER4 (0.51) FFAR1NPC1RAB9AMEN1KMT2A
SCHEMBL11282578 0.75 RXRA (0.43) AKR1C3AKR1C2PTGS1L3MBTL1POLB
SCHEMBL1741211 0.75 AKR1C3 (0.58) AKR1C3AKR1C2AKR1C1PTGS1L3MBTL1
SCHEMBL7908556 0.74 MAOB (0.56) PTGS1L3MBTL1FFAR1LMNA
SCHEMBL22095156 0.73 AKR1C3 (0.73) AKR1C3AKR1C2AKR1C1PTGS1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0118867-A2 Substituted 4,10-dihydro-10-oxothieno benzoxepins, a method of preparing the same and intermediate thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1984-09-19 EP disclosed