SCHEMBL11114869

SCHEMBL11114869

CC(CCC(=O)O)c1ccc(OCc2ccsc2C(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
FFAR1 O14842 6/20 0.41
FFAR4 Q5NUL3 2/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
ALOX5 P09917 1/20 0.39
LTB4R Q15722 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11112172 0.90 L3MBTL1 (0.42) ALDH1A1TSHRFFAR1FFAR4NPC1
SCHEMBL10988964 0.87 FFAR1 (0.40) ALDH1A1TSHRFFAR1FFAR4NPC1
SCHEMBL11115339 0.86 NPC1 (0.43) ALDH1A1TSHRFFAR1FFAR4NPC1
SCHEMBL10984633 0.80 ALDH1A1 (0.39) ALDH1A1FFAR1NPC1RAB9ARXRA
SCHEMBL11114850 0.78 AKR1C3 (0.47) ALDH1A1TSHRFFAR1NPC1RAB9A
SCHEMBL9870392 0.78 FFAR1 (0.50) ALDH1A1TSHRFFAR1FFAR4ALOX5
SCHEMBL11118801 0.77 KMT2A (0.42) ALDH1A1TSHRNPC1RAB9AKDM4E
SCHEMBL11114853 0.77 LTB4R (0.56) FFAR1FFAR4LTB4R
SCHEMBL8936259 0.76 SLC6A1 (0.51) FFAR1NPC1RAB9AKDM4E
SCHEMBL10985950 0.76 RAB9A (0.42) ALDH1A1TSHRFFAR1FFAR4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0118867-A2 Substituted 4,10-dihydro-10-oxothieno benzoxepins, a method of preparing the same and intermediate thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1984-09-19 EP disclosed