SCHEMBL11115732

SCHEMBL11115732

COc1cc(C(=O)N(C)CCN(C)CC=C(c2ccccc2)c2ccccc2)cc(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 3/20 0.45
MAPK1 P28482 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
SCN1A P35498 1/20 0.44
SCN2A Q99250 1/20 0.44
SCN3A Q9NY46 1/20 0.44
ALDH1A1 P00352 5/20 0.43
OPRM1 P35372 2/20 0.43
OPRD1 P41143 2/20 0.43
NR1I2 O75469 1/20 0.43
CHRM2 P08172 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADRA2B P18089 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRK1 P41145 1/20 0.43
CHRNA4 P43681 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PDE4D Q08499 1/20 0.43
KCNH2 Q12809 1/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11113048 0.82 KDM4E (0.51) MAPK1L3MBTL1ALDH1A1CYP1A2SMN1; SMN2
SCHEMBL7273776 0.81 L3MBTL1 (0.59) MAPK1L3MBTL1SCN1ASCN2ASCN3A
SCHEMBL9750661 0.73 SMN1; SMN2 (0.46) ACKR3L3MBTL1SCN1ASCN2ASCN3A
SCHEMBL9750679 0.72 SCN1A (0.49) MAPK1L3MBTL1SCN1ASCN2ASCN3A
Hydrochloric Acid SCHEMBL9750696 0.71 SCN1A (0.48) MAPK1L3MBTL1SCN1ASCN2ASCN3A
SCHEMBL13219952 0.71 ACKR3 (0.69) ACKR3MAPK1L3MBTL1ALDH1A1TNFRSF1A
SCHEMBL7276036 0.70 KMT2A (0.49) MAPK1L3MBTL1SCN1ASCN2ASCN3A
Benzene SCHEMBL27454328 0.69 SCN1A (0.44) ACKR3MAPK1L3MBTL1SCN1ASCN2A
Hydrochloric Acid SCHEMBL7266825 0.69 KMT2A (0.48) MAPK1SCN1ASCN2ASCN3AALDH1A1
Hydrochloric Acid SCHEMBL9750666 0.69 KMT2A (0.48) MAPK1SCN1ASCN2ASCN3AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041757-B1 ETHYLENDIAMINE DERIVATIVES, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND INTERMEDIATES FOR THEIR PREPARATION Simes S.p.A. (IT) 1984-11-07 EP disclosed