SCHEMBL11113048

SCHEMBL11113048

COc1cc(CN(C)CCN(C)CC=C(c2ccccc2)c2ccccc2)cc(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 2/20 0.51
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
TP53 P04637 1/20 0.45
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
BLM P54132 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
DRD1 P21728 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11115732 0.82 ACKR3 (0.45) KDM4EALDH1A1MAPTTP53MAPK1
SCHEMBL9750739 0.81 SIGMAR1 (0.52) SMN1; SMN2SIGMAR1
SCHEMBL7268018 0.81 KDM4E (0.65) KDM4EALDH1A1GAAMAPTMAPK1
Hydrochloric Acid SCHEMBL11113593 0.80 SIGMAR1 (0.51) ALDH1A1SMN1; SMN2BLMSIGMAR1
SCHEMBL11116163 0.80 ACHE (0.56) SIGMAR1ACHE
SCHEMBL15720901 0.75 KDM4E (0.73) KDM4EALDH1A1GAAMAPTMAPK1
SCHEMBL9750783 0.73 ALDH1A1 (0.51) KDM4EALDH1A1GAAMAPTTP53
SCHEMBL11128142 0.73 SIGMAR1 (0.50) ALDH1A1MEN1KMT2ASMN1; SMN2SIGMAR1
SCHEMBL7265472 0.72 AOC3 (0.51) KDM4EALDH1A1GAAMAPTCYP3A4
SCHEMBL7273776 0.72 L3MBTL1 (0.59) KDM4EALDH1A1GAAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041757-B1 ETHYLENDIAMINE DERIVATIVES, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND INTERMEDIATES FOR THEIR PREPARATION Simes S.p.A. (IT) 1984-11-07 EP disclosed
EP-0041757-A1 Ethylendiamine derivatives, preparation thereof, pharmaceutical compositions containing same and intermediates for their preparation Simes S.p.A. (IT) 1981-12-16 EP disclosed