SCHEMBL1120131

SCHEMBL1120131

CC(C)(C)C1CC(c2nc(C(=O)OC3CCCCC3)cs2)CCN1C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.33
HCRTR2 O43614 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
PIM1 P11309 4/20 0.31
PIM3 Q86V86 4/20 0.31
PIM2 Q9P1W9 4/20 0.31
CYP19A1 P11511 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
CPT2 P23786 1/20 0.31
CPT1A P50416 1/20 0.31
CPT1B Q92523 1/20 0.31
HSD11B1 P28845 2/20 0.31
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1120255 0.84 CASP3 (0.42) SMN1; SMN2NPC1HTTRAB9AKDM4E
SCHEMBL2593942 0.83 SMYD3 (0.33) HCRTR2
SCHEMBL1884435 0.82 FAAH (0.38) HRH3PIM1PIM3PIM2HSD11B1
SCHEMBL1120328 0.82 RAB9A (0.36) HCRTR2SMN1; SMN2HTTRAB9AKDM4E
SCHEMBL18192787 0.79 HCRTR2 (0.31) HCRTR2
SCHEMBL2588097 0.79
SCHEMBL2588101 0.79
SCHEMBL18192790 0.77 MEN1 (0.35) SMN1; SMN2NPC1RAB9AMEN1KMT2A
SCHEMBL1120132 0.77 GPR119 (0.47) KDM4EHPGD
SCHEMBL12074811 0.77 PIM1 (0.39) HRH3SMN1; SMN2NPC1RAB9APIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493886-B1 HETEROARYL PIPERIDINE AND PIPERAZINE DERIVATES BAYER CROPSCIENCE AG (DE) 2014-11-26 EP disclosed
EP-2493886-A1 HETEROARYLPIPERIDINE AND -PIPERAZINE DERIVATIVES Bayer CropScience AG (DE) 2012-09-05 EP disclosed
EP-2280965-B1 THIAZOL-4-CARBOXYLIC ACID ESTERS AND THIOESTERS AS PLANT PROTECTION AGENTS BAYER CROPSCIENCE AG (DE) 2012-08-29 EP disclosed
WO-2011051244-A1 HETEROARYLPIPERIDINE AND -PIPERAZINE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2011-05-05 WO disclosed
EP-2280965-A1 THIAZOL-4-CARBOXYLIC ACID ESTERS AND THIOESTERS AS PLANT PROTECTION AGENTS BAYER CROPSCIENCE AG (DE) 2011-02-09 EP disclosed
WO-2009132785-A1 THIAZOL-4-CARBOXYLIC ACID ESTERS AND THIOESTERS AS PLANT PROTECTION AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT 2009-11-05 WO disclosed