SCHEMBL11208405

SCHEMBL11208405

CCc1ccc2cc1-2.CON(OC)OC

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.37
BRD4 O60885 1/20 0.36
PTPRC P08575 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
HSD17B1 P14061 1/20 0.32
PTPN1 P18031 1/20 0.32
GSTP1 P09211 1/20 0.32
RARA P10276 2/20 0.32
RARB P10826 2/20 0.32
RARG P13631 2/20 0.32
HTT P42858 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
ALDH1A1 P00352 1/20 0.30
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL4590632 0.83
SCHEMBL28668871 0.80 TRPA1 (0.37) TRPA1BRD4PTPRCPDCD1CD274
SCHEMBL14134813 0.68 KDM4E (0.44) PTPRCHSD17B1PTPN1KMT2AALDH1A1
Ammonia Solution, Strong SCHEMBL4591099 0.66 ALOX5 (0.46) BRD4RARARARBRARG
SCHEMBL5551523 0.64 BACE1 (0.51) PTPN1HTTMEN1KMT2AALDH1A1
Ammonia Solution, Strong SCHEMBL4604807 0.64
SCHEMBL9516471 0.64 HSD17B1 (0.38) TRPA1PTPRCHSD17B1ALOX5APFEN1
SCHEMBL3921828 0.64 ALDH1A1 (0.55) MEN1KMT2AALDH1A1GAA
SCHEMBL9289360 0.63 L3MBTL1 (0.50) TRPA1PTPRCPDCD1CD274PTPN1
SCHEMBL10916725 0.63 HSD17B1 (0.45) HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105481850-A Tetrahydroberberine derivative and application thereof CHENGDU BASS KERRY BIOLOGICAL TECH CO LTD 2016-04-13 CN disclosed
CN-102516042-A Method for synthesizing 3,4,5-trimethoxylbenzyl chloride TAICANG YUNTONG CHEMICAL FACTORY 2012-06-27 CN disclosed
EP-0028279-B1 PHTHALIDE-ISOQUINOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN MEDICAMENTS CALAIRE CHIMIE S.A. (FR) 1983-02-16 EP disclosed
EP-0028279-A1 Phthalide-isoquinoline derivatives, their preparation and their use in medicaments CALAIRE CHIMIE S.A. (FR) 1981-05-13 EP disclosed