SCHEMBL11224516

SCHEMBL11224516

N#Cc1cccc(Cl)c1C1C(=O)CCCC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 4/20 0.41
LDHB P07195 4/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
CASP1 P29466 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRIA1 P42261 1/20 0.36
CACNG8 Q8WXS5 1/20 0.36
HSD11B1 P28845 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
DYRK1A Q13627 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11217137 0.78 GPR35 (0.38) KDM4EKMT2AMEN1MAPTSMN1; SMN2
SCHEMBL11228339 0.76 LDHA (0.40) LDHALDHBKDM4EALDH1A1GAA
SCHEMBL28032574 0.73 LDHA (0.43) LDHALDHBKDM4EALDH1A1GAA
SCHEMBL11231609 0.72 ABCC9 (0.34) CA1CA2
SCHEMBL11224539 0.72 CRHBP (0.43)
SCHEMBL11226368 0.71 ALDH1A1 (0.41) KDM4EALDH1A1GAAKMT2AMEN1
SCHEMBL10736168 0.67 TP53 (0.47) KDM4EALDH1A1GAAKMT2AMAPT
SCHEMBL15001063 0.65 CRHBP (0.45) HPGDSMN1; SMN2
SCHEMBL989338 0.64 DYRK1A (0.44) KDM4EALDH1A1GAAKMT2AMEN1
SCHEMBL11227905 0.64 CYP3A4 (0.39) KDM4EALDH1A1GAAALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007243-B1 2-ARYL-1,3-CYCLOHEXANEDIONE COMPOUNDS AND ALKALI METAL SALTS, AMMONIUM SALTS AND ENOL ESTERS THEREOF, COMPOSITION AND METHOD OF CONTROLLING ACARINA ECTOPARASITES ON WARMBLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1982-11-17 EP disclosed
US-4257858-A REACTING A CYCLOHEXA-1,3-DIONE-2-DIAZIDE WITH AN ARYL COMPOUND UNION CARBIDE CORPORATION (US) 1981-03-24 US disclosed
US-4256657-A CYCLIZATION, ACID CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256658-A CYCLIZATION, BASIC CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256659-A Method of preparing 2-aryl-1,3-cyclohexanedione compounds UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4209532-A Biocidal 2-aryl-1,3-cyclohexane dione compounds and alkali metal and ammonium salts thereof UNION CARBIDE CORPORATION (US) 1980-06-24 US disclosed
EP-0007243-A1 2-Aryl-1,3-cyclohexanedione compounds and alkali metal salts, ammonium salts and enol esters thereof, composition and method of controlling acarina ectoparasites on warmblooded animals UNION CARBIDE CORPORATION (US) 1980-01-23 EP disclosed
US-4175135-A Method of controlling acarina ectoparasites on warmblooded animals by orally administering to the animal an ectoparasitically effective amount of a 2-aryl-1,3-cyclohexanedione compound, and alkali metal salts, ammonium salts and enol esters thereof UNION CARBIDE CORPORATION (US) 1979-11-20 US disclosed