SCHEMBL11226286

SCHEMBL11226286

CCN1CCCC(c2cccc3[nH]ccc23)C1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
PDE2A O00408 1/20 0.44
ADRA1A P35348 1/20 0.43
HTR1A P08908 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ATM Q13315 1/20 0.42
ADRA1D P25100 2/20 0.41
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11219877 0.90 DRD2 (0.52) DRD2DRD3
SCHEMBL11226328 0.84 KDM4E (0.57) DRD2DRD3ADRA1AHTR1AKDM4E
SCHEMBL10959130 0.84 JAK2 (0.56) DRD2DRD3PDE2AOPRM1OPRK1
SCHEMBL14027792 0.78 HTR1A (0.47) ADRA1AHTR1A
SCHEMBL8995183 0.77 HTR1A (0.48) ADRA1AHTR1AADRA1D
SCHEMBL17429447 0.75 HTR1A (0.51) ADRA1AHTR1A
SCHEMBL3682166 0.75 KDM4E (0.55) ADRA1AHTR1AKDM4EATMADRA1D
SCHEMBL11065117 0.74 BTK (0.45) ADRA1AHTR1AKDM4E
SCHEMBL19210848 0.74 KDM4E (0.70) KDM4EATMADRA1DCYP2D6
SCHEMBL18089303 0.72 DRD2 (0.48) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4332808-A Dopaminergically stimulating 4-substituted indoles ROUSSEL UCLAF (FR) 1982-06-01 US claimed
US-4332808-A Dopaminergically stimulating 4-substituted indoles ROUSSEL UCLAF (FR) 1982-06-01 US disclosed