SCHEMBL11226328

SCHEMBL11226328

CN1CCCC(c2cccc3[nH]ccc23)C1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
ATM Q13315 1/20 0.57
DRD2 P14416 2/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
KCNH2 Q12809 1/20 0.48
HTR1A P08908 1/20 0.44
ADRA1A P35348 1/20 0.43
PARP1 P09874 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11219877 0.84 DRD2 (0.52) DRD2DRD3
SCHEMBL11226286 0.84 DRD2 (0.44) KDM4EATMDRD2HTR1AADRA1A
SCHEMBL3682166 0.82 KDM4E (0.55) KDM4EATMHTR2AHTR1AADRA1A
SCHEMBL10212688 0.82 KDM4E (0.84) KDM4EATMDRD2HTR2AHTR2C
SCHEMBL14027792 0.80 HTR1A (0.47) HTR2CHTR1AADRA1A
SCHEMBL8995183 0.79 HTR1A (0.48) HTR2CHTR1AADRA1A
SCHEMBL10959130 0.78 JAK2 (0.56) DRD2HTR2AHTR2CKCNH2DRD3
SCHEMBL17429447 0.77 HTR1A (0.51) HTR2CHTR1AADRA1A
SCHEMBL21369339 0.77 DRD2 (0.55) KDM4EATMDRD2HTR2AHTR2C
SCHEMBL11065117 0.76 BTK (0.45) KDM4EHTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4332808-A Dopaminergically stimulating 4-substituted indoles ROUSSEL UCLAF (FR) 1982-06-01 US claimed
EP-0021924-A2 Indole derivatives, process for their preparation, their use as medicines and pharmaceutical compositions containing them ROUSSEL-UCLAF (FR) 1981-01-07 EP claimed
US-4332808-A Dopaminergically stimulating 4-substituted indoles ROUSSEL UCLAF (FR) 1982-06-01 US disclosed