SCHEMBL11235898

SCHEMBL11235898

CC(=O)Nc1cc(-c2cc(C)cc(C)n2)c(C)[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
ADORA2A P29274 2/20 0.35
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR3 P22607 1/20 0.35
DYRK1A Q13627 1/20 0.35
PIK3CG P48736 1/20 0.35
DHODH Q02127 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
POLB P06746 1/20 0.33
CCNE2 O96020 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11233196 0.77 KDM4E (0.51) KDM4EGAADYRK1ADHODHPOLB
SCHEMBL11238700 0.76 POLB (0.39) KDM4EGAADHODHCYP1A2POLB
SCHEMBL11232487 0.75 JAK1 (0.46) KDM4EALDH1A1
SCHEMBL11243686 0.75 KDM4E (0.36) KDM4ECYP1A2POLBALDH1A1
SCHEMBL11231843 0.75 PDE3B (0.51) KDM4EGAAFGFR1FGFR2CYP2C19
SCHEMBL10980606 0.74 ADORA2B (0.42) KDM4EADORA2AADORA3CYP2C19CDK2
SCHEMBL10982470 0.74 DRD1 (0.39) KDM4EGAACYP2C9CCNE2CCNE1
SCHEMBL11238639 0.73 PDE3B (0.57) KDM4EGAAADORA2AADORA3CYP2C19
SCHEMBL11235309 0.72 ALDH1A1 (0.58) KDM4EGAAPOLBALDH1A1
SCHEMBL11232009 0.71 KDM4E (0.61) KDM4EGAACYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed