SCHEMBL1124331

SCHEMBL1124331

Cc1ccccc1C=CC(N)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
TSHR P16473 2/20 0.48
RAB9A P51151 3/20 0.47
LMNA P02545 3/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PTPN1 P18031 2/20 0.46
MAPT P10636 1/20 0.44
KDM4E B2RXH2 3/20 0.43
GMNN O75496 1/20 0.43
PMP22 Q01453 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NFE2L2 Q16236 2/20 0.42
NFKB1 P19838 2/20 0.42
JUN P05412 1/20 0.42
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
TFEB P19484 1/20 0.42
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30560932 1.00 ALDH1A1 (0.48) ALDH1A1TSHRRAB9ALMNAHPGD
SCHEMBL1124329 1.00 ALDH1A1 (0.48) ALDH1A1TSHRRAB9ALMNAHPGD
SCHEMBL28358892 1.00 ALDH1A1 (0.48) ALDH1A1TSHRRAB9ALMNAHPGD
SCHEMBL2328371 0.85 NFKB1 (0.50) LMNAHTTPTPN1MAPTKDM4E
SCHEMBL30560977 0.85 PTPN1 (0.40) ALDH1A1TSHRRAB9ALMNAHPGD
SCHEMBL5598954 0.83 NFE2L2 (0.61) ALDH1A1TSHRRAB9ALMNAMAPT
SCHEMBL5598952 0.83 NFE2L2 (0.61) ALDH1A1TSHRRAB9ALMNAMAPT
SCHEMBL17095076 0.83 CD44 (0.41) ALDH1A1TSHRRAB9ALMNAHPGD
SCHEMBL78556 0.82 CA1 (0.62) ALDH1A1TSHRRAB9ALMNAHTT
SCHEMBL2425317 0.82 CA1 (0.62) ALDH1A1TSHRRAB9ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP claimed
WO-2009141782-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2009-11-26 WO claimed
CN-110818584-B Method for synthesizing alpha, beta-unsaturated amide compound by visible light catalysis 闽南师范大学 2023-05-09 CN disclosed
CN-115322131-A Synthesis method of beta-fluoroindole acrylamide compound 温州大学 2022-11-11 CN disclosed
CN-110818584-A Method for synthesizing α -unsaturated amide compound by visible light catalysis 闽南师范大学 2020-02-21 CN disclosed
CN-102898408-B Benzopyran compounds, preparation method and applications thereof SHANGHAI RUIGUANG BIOCHEMICAL SCIENCE AND TECHNOLOGY DEV CO LTD 2015-04-29 CN disclosed
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP disclosed
WO-2009141782-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2009-11-26 WO disclosed
EP-1896417-A1 LINEAR UREA MIMICS ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS Brystol-Myers Squibb Company (US) 2008-03-12 EP disclosed
WO-2007002584-A1 LINEAR UREA MIMICS ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
EP-0737896-B1 Photosensitive composition and photosensitive planographic printing plate KODAK POLYCHROME GRAPHICS JP (JP) 2003-08-27 EP disclosed
US-5731127-A WEAR RESISTANCE, SOLVENT RESISTANCE DAINIPPON INK AND CHEMICALS, INC. (JP) 1998-03-24 US disclosed
EP-0702673-B1 BENZ(B)AZEPINE-2,5-DIONES USEFUL IN THE TREATMENT OF NEURODEGENERATIVE DISORDERS ZENECA LTD (GB) 1998-02-25 EP disclosed
EP-0737896-A2 Photosensitive composition and photosensitive planographic printing plate DAINIPPON INK AND CHEMICALS, INC. (JP) 1996-10-16 EP disclosed