SCHEMBL11246657

SCHEMBL11246657

COc1ccc2sc3cc(CC(=O)O)ccc3c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 2/20 0.58
PTGS1 P23219 1/20 0.58
AKR1C3 P42330 1/20 0.58
KDM4E B2RXH2 5/20 0.46
ALDH1A1 P00352 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
MAPT P10636 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
POLB P06746 1/20 0.45
GAA P10253 3/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 1/20 0.44
NFKB1 P19838 1/20 0.44
PTPN7 P35236 1/20 0.44
DUSP3 P51452 1/20 0.44
PTPN12 Q05209 1/20 0.44
PTPN22 Q9Y2R2 1/20 0.44
LCK P06239 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11248851 0.93 AKR1C2 (0.63) AKR1C2PTGS1AKR1C3KDM4EALDH1A1
SCHEMBL11243330 0.83 SLC22A12 (0.45) KDM4EALDH1A1TDP1MAPTPOLB
SCHEMBL11240186 0.82 EDNRA (0.52) PTPN7DUSP3PTPN12PTPN22PPARG
SCHEMBL11237206 0.82 KDM4E (0.47) AKR1C2PTGS1AKR1C3KDM4EALDH1A1
SCHEMBL11246646 0.80 CA2 (0.49) KDM4EALDH1A1TDP1MAPTPOLB
SCHEMBL11253323 0.80 CYP1A2 (0.47) AKR1C2PTGS1AKR1C3KDM4EALDH1A1
SCHEMBL11240017 0.79 KEAP1 (0.51) KDM4EALDH1A1TDP1MAPTPOLB
SCHEMBL11246422 0.79 KDM4E (0.44) AKR1C2PTGS1AKR1C3KDM4EALDH1A1
SCHEMBL11244551 0.79 KDM4E (0.44) KDM4EALDH1A1TDP1MAPTPOLB
SCHEMBL11243026 0.78 KDM4E (0.41) AKR1C2PTGS1AKR1C3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed