SCHEMBL11248851

SCHEMBL11248851

COc1ccc2c(c1)sc1cc(CC(=O)O)ccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 2/20 0.63
PTGS1 P23219 1/20 0.63
AKR1C3 P42330 1/20 0.63
KDM4E B2RXH2 4/20 0.49
GAA P10253 3/20 0.49
ALDH1A1 P00352 2/20 0.49
TSHR P16473 2/20 0.49
MAPT P10636 2/20 0.49
LMNA P02545 1/20 0.49
PRNP P04156 1/20 0.49
MAPK1 P28482 1/20 0.49
PPARG P37231 1/20 0.49
HTT P42858 1/20 0.49
MAPK10 P53779 1/20 0.49
NCOA2 Q15596 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
POLB P06746 1/20 0.48
HSD17B10 Q99714 1/20 0.48
NFKB1 P19838 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11246657 0.93 AKR1C2 (0.58) AKR1C2PTGS1AKR1C3KDM4EGAA
SCHEMBL11246405 0.81 BCL2L1 (0.50) AKR1C2PTGS1AKR1C3KDM4EGAA
SCHEMBL11232390 0.78 AKR1B1 (0.53) PTGS1KDM4EGAAALDH1A1TSHR
6-Methoxy-2-Naphthylacetic Acid SCHEMBL253759 0.78 AKR1C3 (1.00) AKR1C2PTGS1AKR1C3KDM4EGAA
SCHEMBL11243330 0.78 SLC22A12 (0.45) KDM4EGAAALDH1A1TSHRMAPT
SCHEMBL28654017 0.78 TUBB4A (0.64) MAPTTDP1L3MBTL1
SCHEMBL11242088 0.77 BCKDK (0.51) KDM4EGAAALDH1A1TSHRMAPT
Methane SCHEMBL11248449 0.77 AKR1B1 (0.51) PTGS1KDM4EGAAALDH1A1TSHR
SCHEMBL11425132 0.77 PTGS1 (0.63) AKR1C2PTGS1AKR1C3KDM4EGAA
SCHEMBL11237206 0.77 KDM4E (0.47) AKR1C2PTGS1AKR1C3KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed