SCHEMBL11248814

SCHEMBL11248814

Cc1ccc(F)cc1NC(=N)NC(=O)NC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.47
HTT P42858 2/20 0.47
ALDH1A1 P00352 4/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
IDH1 O75874 1/20 0.42
LMNA P02545 2/20 0.41
PKM P14618 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ESR1 P03372 1/20 0.40
MAPK1 P28482 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
ACKR3 P25106 1/20 0.39
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052569 0.89 ALDH1A1 (0.43) MAPTHTTALDH1A1KDM4EIDH1
SCHEMBL11053888 0.87 HTT (0.47) MAPTHTTALDH1A1LMNAPKM
SCHEMBL11261823 0.85 TAS2R14 (0.44) MAPTHTTALDH1A1IDH1KMT2A
SCHEMBL11263600 0.85 GAA (0.48) MAPTHTTALDH1A1LMNANPSR1
SCHEMBL11258056 0.85 MEN1 (0.47) MAPTHTTALDH1A1HPGDKDM4E
SCHEMBL11054561 0.84 HTT (0.50) MAPTHTTALDH1A1KDM4ELMNA
SCHEMBL11052091 0.82 NPC1 (0.40) MAPTHTTALDH1A1KDM4EPKM
SCHEMBL11053772 0.82 HTT (0.38) MAPTHTTPKMMAPK1KMT2A
SCHEMBL11250897 0.82 PKM (0.48) MAPTHTTPKMKMT2AMEN1
SCHEMBL11052904 0.82 HTT (0.47) HTTMAPK1NPSR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed