SCHEMBL11248847

SCHEMBL11248847

CC(=O)N1CCC(OC(=O)O)(c2ccccc2Sc2ccc(F)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 1/20 0.41
ALDH1A1 P00352 7/20 0.40
LMNA P02545 4/20 0.40
SLC6A9 P48067 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
USP2 O75604 2/20 0.38
MAPK1 P28482 2/20 0.38
CYP2C19 P33261 2/20 0.38
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
GAA P10253 1/20 0.37
GFER P55789 1/20 0.37
CYP2D6 P10635 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.36
ALOX12 P18054 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11257928 0.92 ALDH1A1 (0.46) ALDH1A1LMNASMN1; SMN2USP2MAPK1
SCHEMBL11248413 0.89 SLC6A9 (0.43) ALDH1A1LMNASLC6A9SMN1; SMN2MAPK1
SCHEMBL11248843 0.83 ALDH1A1 (0.42) ITGALALDH1A1LMNASLC6A9SMN1; SMN2
SCHEMBL11249100 0.82 HTR1A (0.43) ALDH1A1LMNASLC6A9MAPK1CYP2D6
Bromide SCHEMBL11248578 0.81 HTR1A (0.43) ALDH1A1LMNASLC6A9MAPK1CYP2D6
SCHEMBL11241295 0.80 USP2 (0.40) ALDH1A1USP2MAPK1CYP2C19MEN1
SCHEMBL11258118 0.78 SLC6A9 (0.43) ALDH1A1LMNASLC6A9SMN1; SMN2MAPK1
SCHEMBL11483416 0.75 ALDH1A1 (0.46) ALDH1A1LMNASMN1; SMN2USP2MAPK1
SCHEMBL11243000 0.75 USP2 (0.43) ALDH1A1LMNAUSP2MAPK1CYP2C19
SCHEMBL11257926 0.74 ALDH1A1 (0.48) ALDH1A1LMNASMN1; SMN2USP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0013424-B1 SPIRO(DIBENZO(B,F)THIEPINE-PIPERIDINES), INTERMEDIATE PRODUCTS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-17 EP disclosed
EP-0013424-A1 Spiro(dibenzo(b,f)thiepine-piperidines), intermediate products for their preparation and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1980-07-23 EP disclosed