SCHEMBL11248413

SCHEMBL11248413

CN1CCC(OC(=O)O)(c2ccccc2Sc2ccc(F)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 4/20 0.43
KDM4E B2RXH2 5/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NPY1R P25929 1/20 0.43
NPY2R P49146 1/20 0.43
ALDH1A1 P00352 4/20 0.42
MAPT P10636 2/20 0.42
OPRM1 P35372 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
GLA P06280 1/20 0.37
HTR1A P08908 1/20 0.37
HTR3A P46098 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
CHRNA7 P36544 1/20 0.36
LMNA P02545 2/20 0.35
SCN1A P35498 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN3A Q9NY46 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11248847 0.89 ITGAL (0.41) SLC6A9SMN1; SMN2ALDH1A1L3MBTL1GLA
SCHEMBL11258118 0.89 SLC6A9 (0.43) SLC6A9KDM4ESMN1; SMN2NPY1RNPY2R
SCHEMBL11249100 0.84 HTR1A (0.43) SLC6A9KDM4EALDH1A1MAPTOPRM1
Bromide SCHEMBL11248578 0.83 HTR1A (0.43) SLC6A9KDM4EALDH1A1MAPTOPRM1
SCHEMBL11248404 0.82 SMN1; SMN2 (0.43) SLC6A9KDM4ESMN1; SMN2NPY1RNPY2R
SCHEMBL11257928 0.80 ALDH1A1 (0.46) KDM4ESMN1; SMN2NPY1RNPY2RALDH1A1
SCHEMBL11255005 0.79 SCN1A (0.41) KDM4ESMN1; SMN2ALDH1A1MAPTOPRM1
SCHEMBL11253112 0.74 HTR1A (0.40) SLC6A9KDM4ESMN1; SMN2NPY1RNPY2R
SCHEMBL11247836 0.74 OPRM1 (0.42) ALDH1A1OPRM1HTR1AHTR3ACHRNA7
Bromide SCHEMBL11247256 0.73 HTR1A (0.40) SLC6A9KDM4ESMN1; SMN2NPY1RNPY2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0013424-B1 SPIRO(DIBENZO(B,F)THIEPINE-PIPERIDINES), INTERMEDIATE PRODUCTS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-17 EP disclosed
EP-0013424-A1 Spiro(dibenzo(b,f)thiepine-piperidines), intermediate products for their preparation and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1980-07-23 EP disclosed