SCHEMBL11249100

SCHEMBL11249100

O=C(O)OC1(c2ccccc2Sc2ccc(F)cc2)CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.43
HTR3A P46098 9/20 0.43
SLC6A9 P48067 3/20 0.40
ALDH1A1 P00352 2/20 0.38
GLA P06280 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPK1 P28482 1/20 0.36
RHEB Q15382 1/20 0.36
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
DPP4 P27487 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL11248578 0.99 HTR1A (0.43) HTR1AHTR3ASLC6A9ALDH1A1GLA
SCHEMBL11253112 0.91 HTR1A (0.40) HTR1AHTR3ASLC6A9ALDH1A1L3MBTL1
Bromide SCHEMBL11247256 0.90 HTR1A (0.40) HTR1AHTR3ASLC6A9ALDH1A1L3MBTL1
SCHEMBL11248413 0.84 SLC6A9 (0.43) HTR1AHTR3ASLC6A9ALDH1A1GLA
SCHEMBL11248847 0.82 ITGAL (0.41) HTR1AHTR3ASLC6A9ALDH1A1GLA
SCHEMBL11249097 0.81 HTR1A (0.46) HTR1AHTR3ASLC6A9ALDH1A1GLA
Bromide SCHEMBL11427938 0.81 HTR1A (0.45) HTR1AHTR3ASLC6A9ALDH1A1GLA
SCHEMBL4702082 0.78 HTR1A (0.50) HTR1AHTR3ASLC6A9ALDH1A1GLA
SCHEMBL11239682 0.78 SLC6A2 (0.44) HTR1AALDH1A1L3MBTL1MAPK1SIGMAR1
Bromide SCHEMBL11242341 0.77 SLC6A2 (0.43) HTR1AALDH1A1L3MBTL1MAPK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0013424-B1 SPIRO(DIBENZO(B,F)THIEPINE-PIPERIDINES), INTERMEDIATE PRODUCTS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-17 EP disclosed
EP-0013424-A1 Spiro(dibenzo(b,f)thiepine-piperidines), intermediate products for their preparation and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1980-07-23 EP disclosed