SCHEMBL11258136

SCHEMBL11258136

COc1cc2c(cc1OC)C(C)(c1ccncc1)OCC2

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.42
CYP11B2 P19099 3/20 0.42
CYP11B1 P15538 2/20 0.42
CYP19A1 P11511 3/20 0.40
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
MAPT P10636 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
PDE10A Q9Y233 1/20 0.34
PARP1 P09874 1/20 0.34
NPC1 O15118 1/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11427100 0.86 PARP1 (0.41) CYP3A4KMT2AMEN1MAPTALDH1A1
SCHEMBL11271602 0.82 PARP1 (0.40) KMT2AMEN1MAPTALDH1A1HPGD
SCHEMBL11668348 0.74 ALDH1A1 (0.39) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL11221731 0.69 ALOX15 (0.39) CYP3A4KMT2AMEN1MAPTALDH1A1
SCHEMBL7289989 0.67 MAOA (0.38) TSHR
SCHEMBL11229451 0.66 ALDH1A1 (0.33) CYP3A4KMT2AMEN1MAPTALDH1A1
SCHEMBL16931627 0.66 MAPT (0.46) CYP3A4CYP11B2CYP11B1MAPTSMN1; SMN2
SCHEMBL11219802 0.65 MAPT (0.33) CYP3A4KMT2AMEN1MAPTALDH1A1
SCHEMBL11674029 0.65 HTT (0.42) KMT2AMEN1MAPTSMN1; SMN2ALDH1A1
SCHEMBL11668352 0.65 SIGMAR1 (0.40) CYP3A4KMT2AMAPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4223151-A 4-(6,7-DIMETHOXY-1-METHYL-ISOCHROMAN-1-YL)PYRIDINE AMERICAN HOME PRODUCTS CORPORATION (US) 1980-09-16 US claimed
US-4351942-A Isochromans AMERICAN HOME PRODUCTS CORP. (US) 1982-09-28 US disclosed
US-4223151-A 4-(6,7-DIMETHOXY-1-METHYL-ISOCHROMAN-1-YL)PYRIDINE AMERICAN HOME PRODUCTS CORPORATION (US) 1980-09-16 US disclosed