SCHEMBL7289989

SCHEMBL7289989

COc1cc2c(cc1OC)C(C)(C1CCNCC1)OCC2

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.38
TSHR P16473 1/20 0.38
TACR1 P25103 2/20 0.37
HTR2A P28223 9/20 0.36
HTR2C P28335 9/20 0.36
HTR2B P41595 9/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11668352 0.75 SIGMAR1 (0.40) MAOATSHRTACR1HTR2AHTR2C
SCHEMBL7292071 0.71 SIGMAR1 (0.49)
SCHEMBL7298566 0.70 SLC6A2 (0.43) TSHR
SCHEMBL7289449 0.69 KCNH2 (0.45) HTR2AHTR2C
SCHEMBL11427100 0.69 PARP1 (0.41) TACR1
SCHEMBL11221731 0.68 ALOX15 (0.39) TACR1
SCHEMBL11668288 0.67 MAOA (0.44) MAOA
SCHEMBL11258136 0.67 CYP3A4 (0.42) TSHR
SCHEMBL11271602 0.65 PARP1 (0.40) TSHRTACR1
SCHEMBL8405226 0.64 MAOA (0.44) MAOATSHRHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458387-B1 Isochromane derivatives AKZO NOBEL NV (NL) 1996-07-03 EP disclosed
US-5393759-A Isochromane derivatives AKZO N.V. (NL) 1995-02-28 US disclosed
US-5238939-A Isochromane derivatives AKZO N.V. (NL) 1993-08-24 US disclosed
EP-0458387-A1 Isochromane derivatives Akzo Nobel N.V. (NL) 1991-11-27 EP disclosed