SCHEMBL11261370

SCHEMBL11261370

CC(=O)NC(=O)CSC(=O)N(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
NPSR1 Q6W5P4 3/20 0.40
ALDH1A1 P00352 6/20 0.39
KMT2A Q03164 4/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.36
CTSK P43235 1/20 0.36
EPHX1 P07099 1/20 0.36
TSHR P16473 2/20 0.35
GPR139 Q6DWJ6 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11264480 0.76 KMT2A (0.60) MTNR1AMTNR1BALDH1A1KMT2APOLB
SCHEMBL11259579 0.73 PAM (0.62) ALDH1A1KMT2AL3MBTL1ATMTDP1
SCHEMBL11264044 0.72 LMNA (0.41) KMT2AMAPTLMNA
SCHEMBL11269396 0.71 LMNA (0.57) MTNR1AMTNR1BALDH1A1KMT2ANPC1
SCHEMBL11267948 0.71 MAPT (0.51) ALDH1A1KMT2ANPC1POLBHTT
SCHEMBL11266403 0.70 CYP1A2 (0.43) ALDH1A1KMT2APOLBHTTMAPT
SCHEMBL11264131 0.70 TDP1 (0.49) ALDH1A1KMT2ANPC1POLBHTT
SCHEMBL11270801 0.70 TDP1 (0.49) ALDH1A1KMT2ANPC1POLBHTT
SCHEMBL10866960 0.69 EPHX1 (0.50) MTNR1AMTNR1BNPSR1ALDH1A1KMT2A
SCHEMBL11277127 0.69 TSHR (0.35) ALDH1A1KMT2AHTTMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4329363-A Substituted mercapto acid amides and their use MERCK & CO., INC. (US) 1982-05-11 US disclosed
US-4216160-A IMMUNOREGULANTS FOR CORRECTING AN INBALANCE OF IMMUNE HOMEOSTASIS MERCK & CO., INC. (US) 1980-08-05 US disclosed
EP-0001989-A1 Substituted mercapto acid amides, process for their preparation, pharmaceutical composition containing same and their use MERCK & CO. INC. (US) 1979-05-30 EP disclosed