SCHEMBL11263009

SCHEMBL11263009

CC(C#N)c1cccc2c(-c3ccc(Br)cc3)nccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
TDO2 P48775 3/20 0.34
PIP4K2A P48426 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ERBB2 P04626 1/20 0.33
IDO1 P14902 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NTRK1 P04629 1/20 0.32
PIM1 P11309 1/20 0.32
ACVR1 Q04771 1/20 0.32
MYC P01106 1/20 0.32
WDR5 P61964 1/20 0.32
LSS P48449 2/20 0.31
CACNA1B Q00975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11260467 0.87 TDO2 (0.42) TDO2ERBB2IDO1KDM4EALDH1A1
SCHEMBL11260894 0.85 SYK (0.34) TDO2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL11260164 0.85 TDO2 (0.33) TDO2ALDH1A1
SCHEMBL11259590 0.78 TRPV1 (0.37) PIK3CAPIK3CBPIK3CGPIP4K2AALDH1A1
SCHEMBL11253329 0.74 TRPV1 (0.44) PIK3CAPIK3CGTDO2IDO1KDM4E
SCHEMBL11261674 0.73 TDO2 (0.36) TDO2PIP4K2AADORA2AADORA1ERBB2
SCHEMBL11267833 0.73 PIP4K2A (0.38) PIP4K2AALDH1A1TRPV1
SCHEMBL11256693 0.72 ALDH1A1 (0.39) TDO2IDO1KDM4EALDH1A1HPGD
SCHEMBL11497570 0.72 ALDH1A1 (0.40) ADORA2AKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL11258335 0.69 ALDH1A1 (0.39) TDO2IDO1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed