SCHEMBL11267833

SCHEMBL11267833

CCC(C(=O)O)c1cccc2c(-c3ccc(Br)cc3)nccc12

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIP4K2A P48426 2/20 0.38
SELPLG Q14242 1/20 0.35
PTGFR P43088 13/20 0.35
CYP3A4 P08684 2/20 0.35
TRPV1 Q8NER1 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11262913 0.86 ALDH1A1 (0.39) SELPLGCYP3A4ALDH1A1CYP1A2
SCHEMBL11259590 0.84 TRPV1 (0.37) PIP4K2ASELPLGCYP3A4TRPV1ALDH1A1
SCHEMBL11261678 0.74 TDP1 (0.45) CYP3A4TRPV1ALDH1A1CYP1A2CYP2C9
SCHEMBL11263009 0.73 PIK3CA (0.35) PIP4K2ATRPV1ALDH1A1
SCHEMBL11256929 0.73 RAB9A (0.40) CYP3A4TRPV1ALDH1A1CYP1A2CYP2C19
SCHEMBL11257836 0.72 BCHE (0.41) DHODH
SCHEMBL11255431 0.72 SELPLG (0.44) SELPLGCYP3A4TRPV1CYP2C9DHODH
SCHEMBL20520340 0.71 PPARG (0.49) ALDH1A1
SCHEMBL11249519 0.71 NPC1 (0.43) CYP3A4TRPV1ALDH1A1CYP1A2CYP2C9
SCHEMBL11253329 0.70 TRPV1 (0.44) CYP3A4TRPV1ALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed