SCHEMBL11263406

SCHEMBL11263406

O=[C]c1cccc(-c2ccc(I)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN5 P54829 1/20 0.36
XDH P47989 1/20 0.36
SLC22A12 Q96S37 1/20 0.36
HSD17B1 P14061 2/20 0.35
HSD17B2 P37059 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
MEN1 O00255 1/20 0.35
ESR1 P03372 1/20 0.35
KMT2A Q03164 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
PGR P06401 3/20 0.35
CA12 O43570 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CHEK1 O14757 1/20 0.33
MGLL Q99685 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
ABL1 P00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97617 0.83 MGLL (0.45) PTPN5XDHSLC22A12MMP12MMP13
SCHEMBL18874455 0.80 CLK4 (0.52) PTPN5XDHSLC22A12MMP12MMP13
SCHEMBL6215483 0.80 GABRG2 (0.45) PTPN5HSD17B1HSD17B2
SCHEMBL2321571 0.80 PTPN5 (0.42) PTPN5XDHSLC22A12HSD17B1HSD17B2
SCHEMBL2322395 0.80 ESR1 (0.61) XDHSLC22A12HSD17B1HSD17B2CYP3A4
SCHEMBL3947358 0.78 MEN1 (0.55) HSD17B1HSD17B2CYP3A4CYP2C9MEN1
SCHEMBL97068 0.76
SCHEMBL2321711 0.76 KIF11 (0.53) PTPN5MGLL
SCHEMBL9321615 0.73 HSD17B1 (0.44) HSD17B1HSD17B2CYP3A4CYP2C9MEN1
SCHEMBL27664209 0.73 MEN1 (0.50) HSD17B1HSD17B2CYP3A4CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4252719-A REMOVAL OF A TERTIARY HYDROGEN FROM A 5-A-STEROID BY CHLORINATING THE STEROID BEING FIRST ESTERIFIED BY AN IODOARYL-CONTAINING ESTERIFICATION AGENT RESEARCH CORPORATION (US) 1981-02-24 US claimed
US-4323512-A Process for the preparation of steroidal 17α-arylcarboxylates SCHERING CORPORATION (US) 1982-04-06 US disclosed