SCHEMBL11266115

SCHEMBL11266115

NNc1nncc(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
HTT P42858 1/20 0.52
IDO1 P14902 1/20 0.47
PIK3CD O00329 1/20 0.46
PIK3CA P42336 1/20 0.46
PIK3CG P48736 1/20 0.46
ATR Q13535 1/20 0.46
XDH P47989 1/20 0.45
CTSS P25774 1/20 0.45
NOTUM Q6P988 1/20 0.43
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
KDM1A O60341 3/20 0.42
MAOB P27338 2/20 0.42
KMO O15229 2/20 0.42
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11510706 0.82 PIK3CD (0.50) IDO1PIK3CDPIK3CAPIK3CGATR
SCHEMBL3398455 0.81 ADORA2A (0.56) MAPTHTTIDO1PIK3CDPIK3CA
SCHEMBL5593110 0.80 AGTR1 (0.68) MAPTIDO1ATRXDHCTSS
SCHEMBL11468072 0.79 KMO (0.58) IDO1PIK3CDPIK3CAPIK3CGXDH
SCHEMBL11160913 0.78 PLK1 (0.45) MAPTIDO1ATRNOTUMADORA2A
SCHEMBL11160970 0.78 AGTR1 (0.48) MAPTIDO1ATRXDHMEN1
SCHEMBL11126066 0.77 MAPT (0.61) MAPTMEN1NPC1KMT2AALDH1A1
SCHEMBL11265993 0.75 F2RL3 (0.47) MAPTIDO1PIK3CDPIK3CAPIK3CG
SCHEMBL11278322 0.75 ALDH1A1 (0.58) MAPTHTTIDO1PIK3CDPIK3CA
SCHEMBL13425801 0.75 MAPT (0.47) MAPTHTTIDO1ATRADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4157392-A HYPOTENSIVE AGENTS, ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS AND NERVOUS SYSTEM EFFECTS DIAMOND SHAMROCK CORPORATION (US) 1979-06-05 US claimed
US-4310551-A Pharmacologically active substituted 1,2,4-triazines DIAMOND SHAMROCK CORPORATION (US) 1982-01-12 US disclosed
US-4251527-A ANTIINFLAMMATORY AGENTS DIAMOND SHAMROCK CORPORATION (US) 1981-02-17 US disclosed
US-4159375-A 6- AND 7-Aryl-1,2,4-triazolo[4,3-b]-1,2,4-triazines AMERICAN CYANAMID COMPANY (US) 1979-06-26 US disclosed
US-4157392-A HYPOTENSIVE AGENTS, ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS AND NERVOUS SYSTEM EFFECTS DIAMOND SHAMROCK CORPORATION (US) 1979-06-05 US disclosed