SCHEMBL11269128

SCHEMBL11269128

O=[N+]([O-])c1cc2c(cc1OCCCN1CCN(c3ccccc3)CC1)CCC2

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
HTR1A P08908 5/20 0.51
DRD3 P35462 4/20 0.51
DRD2 P14416 3/20 0.51
HTR2A P28223 3/20 0.51
HRH1 P35367 3/20 0.51
SIGMAR1 Q99720 3/20 0.51
TMEM97 Q5BJF2 2/20 0.51
HRH3 Q9Y5N1 2/20 0.50
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TDP1 Q9NUW8 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11270784 0.90 KCNH2 (0.53) HTR1ASIGMAR1ALDH1A1KCNH2
SCHEMBL11273991 0.90 DRD2 (0.48) CYP1A2CYP2D6CYP2C19HTR1ADRD3
SCHEMBL11292019 0.81 TSHR (0.59) CYP1A2CYP2D6CYP2C19HTR1ADRD3
SCHEMBL11280762 0.81 DRD3 (0.56) HTR1ADRD3DRD2HTR2AHRH1
SCHEMBL11270622 0.81 DRD3 (0.57) CYP1A2CYP2D6CYP2C19HTR1ADRD3
SCHEMBL11270104 0.81 HTR1A (0.56) CYP1A2CYP2D6CYP2C19HTR1ADRD3
SCHEMBL11266553 0.81 HTR1A (0.62) CYP2D6CYP2C19HTR1ADRD3DRD2
SCHEMBL11301476 0.81 DRD2 (0.53) CYP2D6CYP2C19HTR1ADRD3DRD2
Hydrochloric Acid SCHEMBL11284442 0.80 HTR1A (0.56) CYP1A2CYP2D6CYP2C19HTR1ADRD3
SCHEMBL8687413 0.79 HTR1A (0.49) CYP1A2CYP2D6CYP2C19HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed