SCHEMBL11276199

SCHEMBL11276199

Clc1cccc(N2CCN(CCCOc3cccc4c3CCC4)CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.58
ABCB1 P08183 1/20 0.54
SIGMAR1 Q99720 2/20 0.52
DRD2 P14416 4/20 0.52
DRD4 P21917 1/20 0.52
DRD3 P35462 1/20 0.52
HTR1A P08908 3/20 0.52
HTR2A P28223 3/20 0.52
HTR7 P34969 3/20 0.52
HTR6 P50406 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11275580 0.97 KCNH2 (0.60) KCNH2ABCB1SIGMAR1DRD2DRD4
SCHEMBL11273095 0.89 DRD2 (0.58) SIGMAR1DRD2DRD4DRD3HTR1A
SCHEMBL11279326 0.88 HTR1A (0.63) KCNH2SIGMAR1DRD2DRD3HTR1A
SCHEMBL11301941 0.87 KCNH2 (0.59) KCNH2ABCB1SIGMAR1DRD2HTR1A
SCHEMBL11275248 0.87 HTR1A (0.50) ABCB1SIGMAR1DRD2DRD3HTR1A
SCHEMBL11811688 0.87 DRD2 (0.58) SIGMAR1DRD2DRD4DRD3HTR1A
SCHEMBL11276677 0.86 KCNH2 (0.61) KCNH2ABCB1DRD2DRD3HTR1A
SCHEMBL11275227 0.86 KCNH2 (0.60) KCNH2ABCB1SIGMAR1DRD2DRD4
SCHEMBL11270602 0.86 HTR1A (0.54) SIGMAR1DRD2DRD4DRD3HTR1A
SCHEMBL11809668 0.85 HTR1A (0.63) KCNH2SIGMAR1DRD2DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed