SCHEMBL11279326

SCHEMBL11279326

c1ccc(N2CCN(CCCOc3cccc4c3CCC4)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.63
DRD3 P35462 4/20 0.62
HRH3 Q9Y5N1 4/20 0.62
SIGMAR1 Q99720 3/20 0.58
DRD2 P14416 2/20 0.58
HTR2A P28223 2/20 0.58
HRH1 P35367 2/20 0.58
TMEM97 Q5BJF2 2/20 0.58
KCNH2 Q12809 1/20 0.51
ADRA1A P35348 1/20 0.51
S1PR5 Q9H228 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11809668 0.98 HTR1A (0.63) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11270870 0.96 HTR1A (0.59) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11273977 0.91 HTR1A (0.56) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11273095 0.90 DRD2 (0.58) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11276199 0.88 KCNH2 (0.58) HTR1ADRD3SIGMAR1DRD2HTR2A
SCHEMBL11282809 0.88 HTR1A (0.55) HTR1ADRD3HRH3DRD2HTR2A
SCHEMBL11275248 0.88 HTR1A (0.50) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11811688 0.87 DRD2 (0.58) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11266147 0.87 SLC6A2 (0.55) HTR1ADRD3HRH3SIGMAR1DRD2
SCHEMBL11813710 0.87 HTR1A (0.51) HTR1ADRD3HRH3SIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed