SCHEMBL1127705

SCHEMBL1127705

COCc1cc(-c2ccccc2)c(C(=O)C(=O)O)n1COC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.36
ALDH1A1 P00352 3/20 0.36
HSD17B10 Q99714 2/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
GLA P06280 1/20 0.36
KMT2A Q03164 1/20 0.36
RCE1 Q9Y256 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA3 P34903 1/20 0.35
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
CYP2C19 P33261 1/20 0.34
EGFR P00533 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.33
ASH1L Q9NR48 1/20 0.33
MAPT P10636 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15162338 0.87 ALDH1A1 (0.43) KDM4EALDH1A1HSD17B10GAAMEN1
SCHEMBL1993379 0.85 GABRA1 (0.40) KDM4EALDH1A1GAAGABRA1GABRG2
SCHEMBL15162319 0.80 THRB (0.36) KDM4EALDH1A1HSD17B10GAAMEN1
SCHEMBL15161896 0.68 CNR1 (0.38) KDM4EALDH1A1GABRA1GABRG2GABRB3
SCHEMBL1127378 0.65 HPGD (0.41) ALDH1A1HSD17B10GAASMN1; SMN2MAPT
SCHEMBL1126904 0.64 PPARG (0.35) KDM4EALDH1A1HSD17B10GAAMEN1
SCHEMBL1127123 0.64 ALDH1A1 (0.40) ALDH1A1GAAMEN1KMT2ASMN1; SMN2
SCHEMBL1126951 0.63 CASR (0.39) KDM4EALDH1A1GABRA1GABRG2GABRB3
SCHEMBL24584645 0.63 PGR (0.43) KDM4EALDH1A1GAAMEN1GLA
SCHEMBL31585967 0.63 SMN1; SMN2 (0.39) ALDH1A1HSD17B10MEN1KMT2AGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed