SCHEMBL1127889

SCHEMBL1127889

Cn1c(C(=O)NC(=O)C2(c3ccccc3)CCNCC2)cc(-c2ccc(Cl)cc2Cl)c1-c1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 7/20 0.40
ROCK2 O75116 1/20 0.37
HDAC1 Q13547 1/20 0.36
ESR1 P03372 1/20 0.35
TACR1 P25103 2/20 0.35
SLC6A9 P48067 1/20 0.35
KHK P50053 1/20 0.34
CNR2 P34972 1/20 0.34
AKT1 P31749 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1128119 0.82 CNR1 (0.42) CNR1CNR2
SCHEMBL1848627 0.81 ROCK2 (0.38) CNR1ROCK2HDAC1TACR1CNR2
SCHEMBL1127886 0.76 CNR1 (0.55) CNR1TACR1CNR2
SCHEMBL2570109 0.74 ESR1 (0.51) CNR1ESR1
SCHEMBL476187 0.73 ROCK2 (0.37) CNR1ROCK2HDAC1TACR1CNR2
SCHEMBL1848299 0.73 EP300 (0.47) CNR1ROCK2HDAC1
SCHEMBL1259435 0.71 TACR1 (0.55) CNR1TACR1CNR2
SCHEMBL1850509 0.71 HDAC1 (0.38) CNR1ROCK2HDAC1ESR1TACR1
SCHEMBL476315 0.71 ROCK2 (0.35) CNR1ROCK2HDAC1TACR1CNR2
SCHEMBL2569129 0.70 CNR1 (0.38) CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283008-A2 PYRROLE DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC APPLICATION THEREOF Sanofi-aventis (FR) 2011-02-16 EP disclosed
WO-2009141533-A2 PYRROLE DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC APPLICATION THEREOF SANOFI-AVENTIS (FR) 2009-11-26 WO disclosed