SCHEMBL1129035

SCHEMBL1129035

Cc1cc(C(C)C)c2nc(Cl)[nH]c2c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.35
NUDT1 P36639 1/20 0.35
LMNA P02545 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
CYP1A2 P05177 1/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1128906 0.81 NPC1 (0.33) HTTLMNANPC1RAB9A
SCHEMBL4283192 0.78 ESR1 (0.41) HTTNUDT1NPC1RAB9AHRH4
SCHEMBL1128920 0.74 NPC1 (0.46) NUDT1LMNANPC1RAB9ACYP1A2
SCHEMBL7341936 0.72 ACHE (0.39) HTTNUDT1NPC1RAB9AHRH4
SCHEMBL1128497 0.72 NPC1 (0.45) LMNANPC1RAB9ATRPV1
SCHEMBL1128996 0.68 NPC1 (0.44) LMNANPC1RAB9AHRH4
SCHEMBL13394501 0.67 GAA (0.42) HTTLMNANPC1RAB9AHRH4
SCHEMBL26203737 0.66 GABRA1 (0.42) LMNANOS3NOS1NOS2
SCHEMBL1128775 0.66 LMNA (0.41) LMNANPC1RAB9ATRPV1
SCHEMBL1129053 0.66 NPC1 (0.45) LMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282762-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION Intermune, Inc. (US) 2011-02-16 EP disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed