SCHEMBL11297104

SCHEMBL11297104

Cc1c(C)c(P(c2ccccc2)c2ccccc2)c(P(c2ccccc2)c2ccccc2)c2c1Oc1ccccc1C2

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
MAPKAPK2 P49137 1/20 0.32
DRD1 P21728 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30770347 1.00 MAOA (0.40) MAOAMAOBMAPKAPK2DRD1
SCHEMBL28660534 0.89 MAOA (0.40) MAOAMAOBMAPKAPK2DRD1
SCHEMBL28904464 0.82 NPSR1 (0.32) MAOAMAOB
SCHEMBL6698583 0.77 MAOA (0.52) MAOAMAOBMAPKAPK2
SCHEMBL6599502 0.77 MAOA (0.42) MAOAMAOBMAPKAPK2
SCHEMBL6599506 0.72 MAOA (0.43) MAOAMAOBMAPKAPK2DRD1
SCHEMBL30168142 0.71 MAOA (0.46) MAOAMAOBMAPKAPK2DRD1
SCHEMBL2658102 0.71 MAOA (0.46) MAOAMAOBMAPKAPK2DRD1
SCHEMBL31673358 0.69 MAOA (0.50) MAOAMAOBDRD1
SCHEMBL115187 0.69 MAOA (0.50) MAOAMAOBMAPKAPK2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4746963-A1 MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2026-05-27 EP disclosed
WO-2025082353-A1 POLYMORPHIC FORMS OF THE COMPOUNDS TARGETING MUTANT OF P53 AND USES THEREOF JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2025-04-24 WO disclosed
US-20250051360-A1 SUBSTITUTED HETEROARYL COMPOUND, AND COMPOSITION AND USE THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2025-02-13 US disclosed
WO-2025017045-A1 MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2025-01-23 WO disclosed
US-20240400591-A1 COMPOUNDS TARGETING MUTANT OF P53 JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-12-05 US disclosed
US-20240376075-A1 POLYMORPHIC FORMS OF AURORA A SELECTIVE INHIBITORS AND USES THEREOF JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-11-14 US disclosed
CN-118666870-A Pyrimidopyridine compounds, pharmaceutical compositions and uses thereof 华南理工大学 2024-09-20 CN disclosed
EP-4384510-A1 COMPOUNDS TARGETING MUTANT OF P53 Jacobio Pharmaceuticals Co., Ltd. (CN) 2024-06-19 EP disclosed
WO-2024120471-A1 COMPOUNDS TARGETING MUTANT OF P53 JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-06-13 WO disclosed
WO-2024041503-A1 COMPOUNDS TARGETING Y220C MUTANT OF P53 JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-02-29 WO disclosed
US-9029391-B2 Isoquinoline compounds and methods for treating HIV VIIV HEALTHCARE UK LIMITED (GB) 2015-05-12 US disclosed
US-20140371278-A1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF TIANJIN BINJIANG PHARMA, INC. (CN) 2014-12-18 US disclosed
EP-2804855-A1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF Tianjin Binjiang Pharma, Inc. (CN) 2014-11-26 EP disclosed
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-05 US disclosed
EP-2665724-A1 BICYCLIC INHIBITORS OF ALK AbbVie Inc. (US) 2013-11-27 EP disclosed
US-20130289027-A1 Isoquinoline Compounds And Methods For Treating HIV VIIV HEALTHCARE UK LIMITED (GB) 2013-10-31 US disclosed
WO-2013107283-A1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF TIANJIN BINJIANG PHARMA, INC. (CN) 2013-07-25 WO disclosed
WO-2012142956-A1 PREPARATION METHOD OF TRIFLUOROSTYRENE COMPOUND 中国科学院上海有机化学研究所 (CN) 2012-10-26 WO disclosed
WO-2012102985-A1 ISOQUINOLINE COMPOUNDS AND METHODS FOR TREATING HIV GLAXOSMITHKLINE LLC (US) 2012-08-02 WO disclosed
WO-2012097682-A1 BICYCLIC INHIBITORS OF ALK ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140371278-A1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF CDK2, CDK1, MAP3K1 MAOA 3342/4885MAOB 2698/4885MAPKAPK2 86/4885
US-20240376075-A1 POLYMORPHIC FORMS OF AURORA A SELECTIVE INHIBITORS AND USES THEREOF AURKA, AURKC, AURKB MAOA 1827/4885MAOB 2526/4885MAPKAPK2 1311/4885
US-20240400591-A1 COMPOUNDS TARGETING MUTANT OF P53 TP53, TP53BP1, MDM2 MAOA 4207/4885MAOB 4327/4885MAPKAPK2 716/4885
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ALK, ABL1, BOD1L1 MAOA 729/4885MAOB 293/4885MAPKAPK2 1491/4885
US-20130289027-A1 Isoquinoline Compounds And Methods For Treating HIV MAVS, CCR5, NFATC1 MAOA 2448/4885MAOB 1822/4885MAPKAPK2 3788/4885
US-20250051360-A1 SUBSTITUTED HETEROARYL COMPOUND, AND COMPOSITION AND USE THEREOF TYK2, JAK2, JAK1 MAOA 1895/4885MAOB 1497/4885MAPKAPK2 81/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.