SCHEMBL11345973

SCHEMBL11345973

C=CCC(=O)Cc1ccc(CBr)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
TSHR P16473 2/20 0.33
TRPA1 O75762 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TGM2 P21980 1/20 0.33
CA2 P00918 2/20 0.32
CAMK2A Q9UQM7 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ABCC4 O15439 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9630131 0.85 TGM2 (0.47) CYP1A2CYP2D6MAPK1HSD17B10SMN1; SMN2
SCHEMBL9515186 0.82 CA2 (0.52) CYP1A2CYP2D6MAPK1HSD17B10SMN1; SMN2
SCHEMBL2456680 0.80 CES1 (0.52) CES2CES1MAPK1TSHRALDH1A1
SCHEMBL9339427 0.77 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1CA2LMNAGAA
SCHEMBL8656429 0.77 SMN1; SMN2 (0.55) SMN1; SMN2TSHRALDH1A1TDP1LMNA
SCHEMBL7174072 0.74 KDM4E (0.56) HSD17B10TSHRTRPA1ALDH1A1CA2
SCHEMBL14340616 0.74 TRPA1 (0.44) CES2CES1CYP2D6MAPK1SMN1; SMN2
SCHEMBL14078090 0.74 CES2 (0.44) CES2CES1HSD17B10TSHRTRPA1
SCHEMBL8442271 0.73 CYP3A4 (0.43) CES2CES1MAPK1HSD17B10SMN1; SMN2
SCHEMBL20060326 0.72 ALOX5 (0.34) CYP1A2CYP2D6MAPK1HSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0021636-A1 Secondary amines, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-01-07 EP disclosed