SCHEMBL1134858

SCHEMBL1134858

O=C(NCCc1ccccc1)c1cccc2[nH]ncc12

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.60
RAB9A P51151 4/20 0.60
ALDH1A1 P00352 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
METTL3 Q86U44 10/20 0.55
KDM4E B2RXH2 1/20 0.54
PRMT5 O14744 1/20 0.52
ROCK2 O75116 1/20 0.50
ROCK1 Q13464 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1134947 0.87 METTL3 (0.56) NPC1RAB9AALDH1A1SMN1; SMN2METTL3
SCHEMBL12821441 0.79 ALDH1A1 (0.60) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL459667 0.78 METTL3 (0.52) NPC1RAB9AMETTL3PRMT5
SCHEMBL13073501 0.76 RAB9A (0.63) NPC1RAB9AALDH1A1KDM4E
SCHEMBL305699 0.76 METTL3 (0.55) METTL3PRMT5
SCHEMBL24112335 0.75 METTL3 (0.55) METTL3
SCHEMBL950058 0.75 RAB9A (1.00) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL17738840 0.74 PKM (0.53) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL1134904 0.74 HSP90AA1 (0.59) METTL3
SCHEMBL30285533 0.74 NOS1 (0.52) NPC1RAB9AALDH1A1SMN1; SMN2METTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2285783-A1 INDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2011-02-23 EP disclosed
WO-2009134666-A1 INDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-11-05 WO disclosed