SCHEMBL11392001

SCHEMBL11392001

Cc1cc(C)c(CCC(=O)CCc2c(C)cc(C)cc2C)c(C)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.42
HRH3 Q9Y5N1 3/20 0.42
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
IAPP P10997 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14988768 0.84 NPSR1 (0.57) GPR17HRH3NPSR1KDM4EKMT2A
SCHEMBL11099663 0.84 KDM4E (0.44) GPR17HRH3NPSR1LMNAKDM4E
SCHEMBL6017716 0.84 GPR17 (0.41) GPR17HRH3NPSR1LMNAKDM4E
SCHEMBL7193838 0.81 ALDH1A1 (0.42) GPR17HRH3NPSR1LMNAKDM4E
SCHEMBL27986523 0.79 ALDH1A1 (0.36) NPSR1LMNAALDH1A1KMT2AMEN1
SCHEMBL1697848 0.79 GPR17 (0.39) GPR17HRH3NPSR1LMNAKDM4E
SCHEMBL28030638 0.79 KMT2A (0.46) NPSR1KMT2AIAPPTDP1L3MBTL1
SCHEMBL3670255 0.78 FABP4 (0.50) GPR17NPSR1KDM4EKMT2AMEN1
SCHEMBL2441173 0.78 GPR17 (0.38) GPR17HRH3NPSR1LMNAALDH1A1
SCHEMBL27986393 0.78 ALDH1A1 (0.37) NPSR1LMNAALDH1A1MAPTIAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4260760-A BACTERICIDES, ALGICIDES MERCK & CO., INC. (US) 1981-04-07 US disclosed
US-4172094-A Polyamine compounds MERCK & CO., INC. (US) 1979-10-23 US disclosed
US-4079059-A ANTIMICROBIAL, ALGAE INHIBITORS MERCK & CO., INC. (US) 1978-03-14 US disclosed
US-4070400-A MICROBIOCIDES, ALGICIDES MERCK & CO., INC. (US) 1978-01-24 US disclosed
US-4061775-A Polyamine compounds as antibacterial agents MERCK & CO., INC. (US) 1977-12-06 US disclosed
US-4058624-A Broad spectrum antibacterial compositions containing tris (hydroxymethyl)-aminomethane and diphenyl and loweralkyl substituted diphenyl polyamines MERCK & CO., INC. (US) 1977-11-15 US disclosed