SCHEMBL1143348

SCHEMBL1143348

Nc1nnc(-c2ccc(Cl)cc2)o1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 1.00
NOTUM Q6P988 2/20 1.00
DGAT1 O75907 1/20 0.66
NPC1 O15118 7/20 0.60
RAB9A P51151 7/20 0.60
HSD17B10 Q99714 5/20 0.60
TP53 P04637 3/20 0.60
TSHR P16473 3/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
MAOA P21397 1/20 0.56
MAOB P27338 1/20 0.56
ALDH1A1 P00352 4/20 0.55
NFKB1 P19838 1/20 0.53
CASP3 P42574 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
MAPT P10636 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21887193 0.84 NPC1 (0.79) KDM4ENOTUMNPC1RAB9AHSD17B10
SCHEMBL26673871 0.83 NPC1 (0.78) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL10112953 0.79 KDM4E (0.66) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL12550898 0.79 KDM4E (0.66) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL20767009 0.79 NPC1 (0.72) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL6903361 0.79 KDM4E (1.00) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL15718167 0.79 DGAT1 (1.00) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL11476623 0.79 KDM4E (0.65) KDM4ENOTUMNPC1RAB9AHSD17B10
SCHEMBL10308910 0.79 KDM4E (0.65) KDM4ENOTUMDGAT1NPC1RAB9A
SCHEMBL28273185 0.79 KDM4E (0.65) KDM4ENOTUMDGAT1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122059901-A 1,3, 4-Oxadiazole compound and preparation method and application thereof 成都大学 2026-05-19 CN disclosed
US-20250346588-A1 IMIDAZOPYRIDINE AND OXAZOLOPYRIDINE DERIVATIVES AND ANALOGS THEREOF, METHODS OF PREPARATION THEREOF, METHODS OF HIF-1/2A PATHWAY INHIBITION, AND INDUCTION OF FERROPTOSIS KUDA THERAPEUTICS INC (US) 2025-11-13 US disclosed
US-12459936-B2 Benzamide antibacterial agents PURDUE RESEARCH FOUNDATION (US) 2025-11-04 US disclosed
WO-2025224262-A1 COMBINATION THERAPIES COMPRISING A CDK2 DEGRADER AND A CDK4/6 INHIBITOR MONTE ROSA THERAPEUTICS AG (CH) 2025-10-30 WO disclosed
EP-4608816-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND METHODS OF USE THEREOF Monte Rosa Therapeutics AG (CH) 2025-09-03 EP disclosed
US-20250263395-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND METHODS OF USE THEREOF MONTE ROSA THERAPEUTICS AG (CH) 2025-08-21 US disclosed
EP-4531838-A1 IMIDAZOPYRIDINE AND OXAZOLOPYRIDINE DERIVATIVES AND ANALOGS THEREOF, METHODS OF PREPARATION THEREOF, METHODS OF HIF-1/2A PATHWAY INHIBITION, AND INDUCTION OF FERROPTOSIS Kuda Therapeutics, Inc. (US) 2025-04-09 EP disclosed
WO-2024092039-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND METHODS OF USE THEREOF MONTE ROSA THERAPEUTICS, INC. (US) 2024-05-02 WO disclosed
WO-2023234970-A1 IMIDAZOPYRIDINE AND OXAZOLOPYRIDINE DERIVATIVES AND ANALOGS THEREOF, METHODS OF PREPARATION THEREOF, METHODS OF HIF-1/2A PATHWAY INHIBITION, AND INDUCTION OF FERROPTOSIS KUDA Therapeutics, Inc. (US) 2023-12-07 WO disclosed
US-20230391767-A1 BENZAMIDE ANTIBACTERIAL AGENTS PURDUE RESEARCH FOUNDATION 2023-12-07 US disclosed
EP-2948446-A1 FLUORO-[1,3]OXAZINES AS BACE1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2015-12-02 EP disclosed
US-20150275076-A1 Non-crystallizable Pi-conjugated Molecular Glass Mixtures, Charge Transporting Molecular Glass Mixtures, Luminescent Molecular Glass Mixtures, or Combinations Thereof for Organic Light Emitting Diodes and other Organic Electronics and Photonics Applications Molaire Consulting 2015-10-01 US disclosed
US-20150275076-A1 Non-crystallizable Pi-conjugated Molecular Glass Mixtures, Charge Transporting Molecular Glass Mixtures, Luminescent Molecular Glass Mixtures, or Combinations Thereof for Organic Light Emitting Diodes and other Organic Electronics and Photonics Applications Molaire Consulting 2015-10-01 US disclosed
CN-103980222-A 2-amido-5-substituted-1,3,4-oxadiazole as well as preparation method and application thereof UNIV SHAANXI SCIENCE & TECH 2014-08-13 CN disclosed
WO-2014114532-A1 FLUORO-[1,3]OXAZINES AS BACE1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2014-07-31 WO disclosed
US-20140179735-A1 TYROSINE PHOSPHATASE INHIBITORS AND USES THEREOF TO MODULATE THE ACTIVITY OF ENZYMESp INVOLVED IN THE PATHOLOGY OF MYCOBACTERIUM TUBERCULOSIS INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION 2014-06-26 US disclosed
US-20110190285-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT ABSOLUTE SCIENCE, INC. (US) 2011-08-04 US disclosed
US-20110034521-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-02-10 US disclosed
US-20070244071-A1 Treatment of proliferative diseases MOUNT SINAI HOSPITAL (CA) 2007-10-18 US disclosed
US-20070244071-A1 Treatment of proliferative diseases MOUNT SINAI HOSPITAL (CA) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230391767-A1 BENZAMIDE ANTIBACTERIAL AGENTS HDAC6, HDAC5, HDAC3 KDM4E 1365/4885NOTUM 1685/4885DGAT1 848/4885
US-20250346588-A1 IMIDAZOPYRIDINE AND OXAZOLOPYRIDINE DERIVATIVES AND ANALOGS THEREOF, METHODS OF PREPARATION THEREOF, METHODS OF HIF-1/2A PATHWAY INHIBITION, AND INDUCTION OF FERROPTOSIS HIF1AN, HIF1A, EGLN2 KDM4E 1020/4885NOTUM 4855/4885DGAT1 3995/4885
US-20110034521-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES MMP7, MMP3, MMP9 KDM4E 1274/4885NOTUM 1467/4885DGAT1 1098/4885
US-12459936-B2 Benzamide antibacterial agents HDAC6, HDAC5, HDAC3 KDM4E 1365/4885NOTUM 1685/4885DGAT1 848/4885
US-20140179735-A1 TYROSINE PHOSPHATASE INHIBITORS AND USES THEREOF TO MODULATE THE ACTIVITY OF ENZYMESp INVOLVED IN THE PATHOLOGY OF MYCOBACTERIUM TUBERCULOSIS PPP3CB, PPP4C, PTPRB KDM4E 739/4885NOTUM 1223/4885DGAT1 4072/4885
US-20110190285-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT NPY5R, RAC3, CPA3 KDM4E 1963/4885NOTUM 1463/4885DGAT1 4017/4885
US-20070244071-A1 Treatment of proliferative diseases CCNO, CCNY, CCNI KDM4E 2806/4885NOTUM 3210/4885DGAT1 2772/4885
US-20250263395-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND METHODS OF USE THEREOF CDK2, SKP2, CDK1 KDM4E 2198/4885NOTUM 3561/4885DGAT1 3296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.