SCHEMBL11501658

SCHEMBL11501658

CS(=O)(=O)O.CS(=O)(=O)O.CSCCCNC(=O)N(CCCCCCN(C(=N)N)C(=O)NCCCSC)C(=N)N

nearest known ligand 0.33

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPY1R P25929 1/20 0.33
ALB P02768 1/20 0.33
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
ALOX15 P16050 1/20 0.31
SPHK1 Q9NYA1 3/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11502077 0.94 ALDH1A1 (0.33) NPY1RALBFNTAFNTBSPHK1
SCHEMBL11501597 0.81 KMT2A (0.46) NPY1RALDH1A1
SCHEMBL11501551 0.77 KDM4E (0.33) KDM4ELMNAGAASMN1; SMN2NPY1R
SCHEMBL8032200 0.77 EPHX1 (0.47) SPHK1
SCHEMBL11460240 0.74 USP2 (0.41) KDM4ESPHK1ALDH1A1
SCHEMBL3070903 0.73 EPHX1 (0.40) ALOX15SPHK1
SCHEMBL11501889 0.73 KMT2A (0.47) SMN1; SMN2NPY1RALDH1A1
SCHEMBL11501702 0.72 SPHK1 (0.43) SPHK1
SCHEMBL11501651 0.72 MTNR1A (0.48) SMN1; SMN2ALDH1A1
SCHEMBL11502016 0.70 TSHR (0.35) SMN1; SMN2NPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4163022-A ANTIPLAQUE AGENTS COOPER LABORATORIES, INC. (US) 1979-07-31 US disclosed