SCHEMBL11520909

SCHEMBL11520909

Cc1noc(-c2cccc([N+](=O)[O-])c2)c1C(=O)Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
TSHR P16473 2/20 0.47
PKM P14618 1/20 0.46
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
EDNRA P25101 2/20 0.45
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
EDNRB P24530 1/20 0.43
MAPT P10636 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
CHRNB2 P17787 1/20 0.41
CHRNA5 P30532 1/20 0.41
CHRNA4 P43681 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11517059 0.80 MEN1 (0.55) ALDH1A1TSHRPKMNPC1RAB9A
SCHEMBL4030555 0.79 MAPT (0.47) ALDH1A1PKMNPC1RAB9AEDNRA
SCHEMBL4030546 0.79 MAPT (0.47) ALDH1A1PKMNPC1RAB9AEDNRA
SCHEMBL893014 0.78 PTGS1 (0.51) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL11516385 0.74 GHSR (0.43) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL11520591 0.72 POLB (0.44) ALDH1A1TSHRNPC1RAB9AMEN1
SCHEMBL12465975 0.72 RAB9A (0.49) ALDH1A1NPC1RAB9AEDNRAMEN1
SCHEMBL4034366 0.72 AKR1C3 (0.43) ALDH1A1PKMNPC1RAB9AEDNRA
SCHEMBL11518747 0.71 MAPT (0.51) ALDH1A1PKMNPC1RAB9AMEN1
SCHEMBL20501599 0.71 ALDH1A1 (0.53) ALDH1A1TSHRPKMNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed