SCHEMBL11524635

SCHEMBL11524635

O=C(NC(=O)c1c(C(F)(F)F)cccc1C(F)(F)F)Nc1cnc(Cl)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.43
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
DYRK3 O43781 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
CDK1 P06493 1/20 0.40
CDK2 P24941 1/20 0.40
FLT4 P35916 1/20 0.40
CSNK1D P48730 1/20 0.40
CLK2 P49760 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
LIMK1 P53667 1/20 0.40
CSNK2A1 P68400 1/20 0.40
CDK5 Q00535 1/20 0.40
STK3 Q13188 1/20 0.40
DYRK1A Q13627 1/20 0.40
BRSK1 Q8TDC3 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11519411 0.85 RAB9A (0.47) TYK2NPC1RAB9AKDM4EMAPT
SCHEMBL11523266 0.81 RAB9A (0.45) NPC1RAB9AKDM4EMEN1MAPT
SCHEMBL11523665 0.80 HCRTR1 (0.48) TYK2NPC1RAB9AMAP4K4CSNK2A1
SCHEMBL11521954 0.79 TYK2 (0.44) TYK2NPC1RAB9AKDM4EALDH1A1
SCHEMBL11522756 0.78 KDM4E (0.48) TYK2NPC1RAB9AKDM4EALDH1A1
SCHEMBL11524682 0.76 TYK2 (0.41) TYK2NPC1RAB9AKDM4EALDH1A1
SCHEMBL8657584 0.75 RAB9A (0.57) NPC1RAB9ARPS6KA3MEN1MAPT
SCHEMBL11520381 0.73 NR1H2 (0.45) DYRK3PRKD3MAP4K4CDK1CDK2
SCHEMBL11524433 0.73 MEN1 (0.45) NPC1KDM4EALDH1A1MAPK1RORC
SCHEMBL11524573 0.73 RAB9A (0.46) TYK2NPC1RAB9AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed