SCHEMBL11544146

SCHEMBL11544146

COC(=O)C=C(C)c1ccc(-c2ccc(Br)cc2Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.38
LTB4R Q15722 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
EGFR P00533 1/20 0.36
MAPT P10636 7/20 0.36
ALDH1A1 P00352 4/20 0.36
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
GPR183 P32249 1/20 0.36
KMT2A Q03164 4/20 0.35
HTT P42858 2/20 0.35
MAPK1 P28482 2/20 0.35
PRKCZ Q05513 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11544143 1.00 SLC6A3 (0.38) SLC6A3LTB4RSMN1; SMN2HDAC3HDAC1
SCHEMBL11542478 0.86 NR4A1 (0.45) LTB4RMMP2MMP9MMP8MMP13
SCHEMBL11542474 0.86 NR4A1 (0.45) LTB4RMMP2MMP9MMP8MMP13
SCHEMBL11543256 0.85 F2 (0.38) SMN1; SMN2MAPTALDH1A1RAB9ANPC1
SCHEMBL11543258 0.85 F2 (0.38) SMN1; SMN2MAPTALDH1A1RAB9ANPC1
SCHEMBL22390293 0.83 ALDH1A1 (0.47) SMN1; SMN2MAPTALDH1A1RAB9ANPC1
SCHEMBL22390294 0.83 ALDH1A1 (0.47) SMN1; SMN2MAPTALDH1A1RAB9ANPC1
SCHEMBL11543441 0.79 HSD17B1 (0.51) SMN1; SMN2MAPTRAB9ANPC1KMT2A
SCHEMBL11485877 0.77 MTNR1A (0.40) SMN1; SMN2HDAC1MAPTALDH1A1RAB9A
SCHEMBL11485879 0.77 MTNR1A (0.40) SMN1; SMN2HDAC1MAPTALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4151302-A Araliphatic dihalogen compounds composition and method of use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-04-24 US disclosed
US-4057647-A Araliphatic dihalogen compounds and process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-11-08 US disclosed