SCHEMBL115452

SCHEMBL115452

Cc1nc2cc(N)ccc2o1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 13/20 0.60
NPC1 O15118 12/20 0.60
SMN1; SMN2 Q16637 9/20 0.60
MAPT P10636 8/20 0.60
KDM4E B2RXH2 7/20 0.60
HSD17B10 Q99714 5/20 0.60
ALDH1A1 P00352 5/20 0.60
TP53 P04637 5/20 0.60
L3MBTL1 Q9Y468 3/20 0.60
NFKB1 P19838 1/20 0.60
NFKB2 Q00653 1/20 0.60
RELA Q04206 1/20 0.60
GFER P55789 4/20 0.58
RXFP1 Q9HBX9 2/20 0.58
TSHR P16473 1/20 0.57
GAA P10253 2/20 0.56
HPGD P15428 3/20 0.55
CASP3 P42574 2/20 0.55
SENP8 Q96LD8 1/20 0.55
SENP7 Q9BQF6 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3979439 0.98 RAB9A (0.58) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL615340 0.84 SMN1; SMN2 (0.58) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL17307530 0.83 RAB9A (0.44) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL29442076 0.79 NPC1 (0.61) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL9105844 0.79 NPC1 (0.61) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL13528421 0.79 L3MBTL1 (0.82) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL903255 0.79 NPC1 (0.61) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL6398262 0.79 MAPT (0.66) RAB9ANPC1SMN1; SMN2MAPTKDM4E
SCHEMBL1192928 0.79 RAB9A (0.43) RAB9ANPC1SMN1; SMN2MAPTKDM4E
Iodide SCHEMBL8417295 0.78 NPC1 (0.59) RAB9ANPC1SMN1; SMN2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 162 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3416948-B1 INDACENE BEARING SULFONYLUREAS AS ANTI-INFLAMMATORY AGENTS UNIV QUEENSLAND (AU) 2024-07-24 EP claimed
US-8461159-B2 Heteroaryl-substituted urea modulators of fatty acid amide hydrolase Jannsen Pharmaceutica BV (BE) 2013-06-11 US claimed
WO-2010068453-A1 HETEROARYL-SUBSTITUTED UREA MODULATORS OF FATTY ACID AMIDE HYDROLASE JANSSEN PHARMACEUTICA NV (BE) 2010-06-17 WO claimed
US-12528810-B2 Small molecule inhibitors of DYRK/CLK and uses thereof ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2026-01-20 US disclosed
US-20250051325-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA 2025-02-13 US disclosed
CN-119306712-A Diaryl pyrimidine derivative containing condensed heterocycle and preparation method and application thereof 山东大学 2025-01-14 CN disclosed
WO-2024188086-A1 AROMATIC AMIDE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 浙江海正药业股份有限公司 2024-09-19 WO disclosed
US-12054483-B2 Small molecule inhibitors of DYRK/CLK and uses thereof ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2024-08-06 US disclosed
EP-3246963-B1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO LTD (KR) 2023-05-31 EP disclosed
US-20220153756-A1 ANTI-INFECTIVE COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2022-05-19 US disclosed
US-20220041590-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA 2022-02-10 US disclosed
EP-0294461-B1 SOLID PARTICLE DISPERSION FILTER DYES FOR PHOTOGRAPHIC COMPOSITIONS EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1991-10-23 EP disclosed
US-5055387-A Silver halide emulsion layer containing a merocyanine dye on a support EASTMAN KODAK COMPANY (US) 1991-10-08 US disclosed
EP-0446845-A2 Sensitizing dye for photographic materials EASTMAN KODAK COMPANY (US) 1991-09-18 EP disclosed
US-4940654-A Solid particle dispersion filter dyes for photographic compositions EASTMAN KODAK COMPANY (US) 1990-07-10 US disclosed
US-4900652-A FILM SUPPORT CAPABLE OF TRANSMITTING RADIATION. EASTMAN KODAK COMPANY (US) 1990-02-13 US disclosed
US-4900653-A SOLUBILITY; CYANINE DYES EASTMAN KODAK COMPANY (US) 1990-02-13 US disclosed
EP-0323728-A2 Filter dyes for photographic elements EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1989-07-12 EP disclosed
EP-0294461-A1 SOLID PARTICLE DISPERSION FILTER DYES FOR PHOTOGRAPHIC COMPOSITIONS. EASTMAN KODAK CO (US) 1988-12-14 EP disclosed
WO-1988004794-A1 SOLID PARTICLE DISPERSION FILTER DYES FOR PHOTOGRAPHIC COMPOSITIONS EASTMAN KODAK COMPANY (US) 1988-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12528810-B2 Small molecule inhibitors of DYRK/CLK and uses thereof CLK3, CLK2, CLK1 RAB9A 3245/4885NPC1 3157/4885SMN1; SMN2 3372/4885
US-20220153756-A1 ANTI-INFECTIVE COMPOUNDS RABGGTB, ELANE, SERPINB1 RAB9A 1091/4885NPC1 402/4885SMN1; SMN2 4839/4885
US-20220041590-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF CLK2, CLK1, CLK3 RAB9A 4181/4885NPC1 3961/4885SMN1; SMN2 4476/4885
US-12054483-B2 Small molecule inhibitors of DYRK/CLK and uses thereof CLK2, CLK1, CLK3 RAB9A 4181/4885NPC1 3961/4885SMN1; SMN2 4476/4885
US-20250051325-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF CLK2, CLK1, CLK3 RAB9A 4181/4885NPC1 3961/4885SMN1; SMN2 4476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.