SCHEMBL11545463

SCHEMBL11545463

CCOC(=O)C=C(C)c1ccc(Oc2ccc(Cl)cc2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.48
MAOA P21397 2/20 0.48
P2RX3 P56373 3/20 0.41
CYP11B1 P15538 3/20 0.40
CYP11B2 P19099 3/20 0.40
CYP1A2 P05177 2/20 0.39
ABCB11 O95342 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
HTR2A P28223 1/20 0.39
PMP22 Q01453 1/20 0.39
PPARA Q07869 1/20 0.39
F2 P00734 1/20 0.39
PLG P00747 1/20 0.39
PRSS1 P07477 1/20 0.39
LMNA P02545 2/20 0.39
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11540801 0.86 MAOB (0.48) MAOBMAOAP2RX3CYP11B1CYP11B2
SCHEMBL11544488 0.83 MAOB (0.50) MAOBMAOAP2RX3CYP11B1CYP11B2
SCHEMBL31294436 0.80 CES2 (0.46) MAOBCYP11B1CYP11B2CYP1A2TSHR
SCHEMBL22407068 0.79 MAOB (0.68) MAOBMAOAP2RX3CYP11B1CYP11B2
SCHEMBL11540804 0.78 MAOB (0.47) MAOBMAOAP2RX3CYP11B1CYP11B2
SCHEMBL11545459 0.78 F2 (0.43) F2PLGPRSS1LMNAALDH1A1
SCHEMBL5255602 0.78 MAOB (0.52) MAOBMAOAP2RX3CYP11B1CYP11B2
SCHEMBL2999106 0.76 ALDH1A1 (0.50) CYP3A4TSHRALDH1A1MAPTTHRB
SCHEMBL2999108 0.76 ALDH1A1 (0.50) CYP3A4TSHRALDH1A1MAPTTHRB
SCHEMBL17169101 0.74 KDM4E (0.49) CYP1A2CYP3A4TSHRLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4151302-A Araliphatic dihalogen compounds composition and method of use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-04-24 US disclosed
US-4057647-A Araliphatic dihalogen compounds and process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-11-08 US disclosed