SCHEMBL11540801

SCHEMBL11540801

COC(=O)C=C(C)c1ccc(Oc2ccc(Cl)cc2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.48
MAOA P21397 1/20 0.48
CYP11B1 P15538 4/20 0.43
CYP11B2 P19099 4/20 0.43
P2RX3 P56373 3/20 0.42
LMNA P02545 1/20 0.41
SCN9A Q15858 2/20 0.38
CPS1 P31327 1/20 0.38
PNLIP P16233 2/20 0.38
TLR8 Q9NR97 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
BRAF P15056 1/20 0.37
HDAC1 Q13547 1/20 0.37
SCN8A Q9UQD0 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11544488 0.86 MAOB (0.50) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL11545463 0.86 MAOB (0.48) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL17996051 0.82 P2RX3 (0.55) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL22407068 0.82 MAOB (0.68) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL22406928 0.80 CYP11B1 (0.48) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL11540804 0.78 MAOB (0.47) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL22406882 0.77 MAOB (0.46) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL11540797 0.76 SCN9A (0.46) LMNASCN9ASCN8ASCN10A
SCHEMBL5255602 0.75 MAOB (0.52) MAOBMAOACYP11B1CYP11B2P2RX3
SCHEMBL5260362 0.75 MAOB (0.49) MAOBMAOACYP11B1CYP11B2P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4151302-A Araliphatic dihalogen compounds composition and method of use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-04-24 US disclosed
US-4057647-A Araliphatic dihalogen compounds and process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-11-08 US disclosed