SCHEMBL11547110

SCHEMBL11547110

NC(=O)c1ccc(OCCNCC(O)COc2cccc(O)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 6/20 0.51
ADRB1 P08588 6/20 0.51
ADRB3 P13945 4/20 0.51
CYP1A2 P05177 1/20 0.51
ATM Q13315 1/20 0.49
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 2/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HSD17B10 Q99714 2/20 0.44
ABCB1 P08183 3/20 0.43
PARP10 Q53GL7 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAPK1 P28482 1/20 0.42
HPGD P15428 1/20 0.42
PMP22 Q01453 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11547838 0.81 ADRB1 (0.56) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11548581 0.80 ADRB1 (0.49) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11549418 0.79 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11549141 0.78 ATM (0.53) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11545485 0.77 ADRB2 (0.51) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11543785 0.77 ADRB2 (0.56) ADRB2ADRB1ADRB3CYP1A2ATM
Tolamolol SCHEMBL613511 0.77 ATM (0.59) ADRB2ADRB1ADRB3CYP1A2ATM
Tolamolol SCHEMBL611643 0.77 ATM (0.59) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11545209 0.76 ATM (0.53) ADRB2ADRB1ADRB3CYP1A2ATM
SCHEMBL11884013 0.76 ADRB1 (0.49) ADRB2ADRB1ADRB3CYP1A2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed