SCHEMBL11554602

SCHEMBL11554602

Oc1cc(C2CNCCN2)cc(O)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.41
QDPR P09417 1/20 0.34
DRD1 P21728 10/20 0.33
KDM4E B2RXH2 7/20 0.33
DRD2 P14416 6/20 0.33
RECQL P46063 4/20 0.33
MAPT P10636 4/20 0.33
BLM P54132 3/20 0.33
CYP3A4 P08684 3/20 0.33
NFKB1 P19838 3/20 0.33
THPO P40225 3/20 0.33
HIF1A Q16665 3/20 0.33
HSD17B10 Q99714 3/20 0.33
DRD5 P21918 3/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP1A2 P05177 1/20 0.33
PKM P14618 1/20 0.33
MTOR P42345 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11553565 0.81 QDPR (0.51) QDPRDRD1KDM4EDRD2MAPT
SCHEMBL6131967 0.74 ESR2 (0.38) DRD1KDM4EDRD2RECQLMAPT
SCHEMBL14258976 0.74 BMPR1B (0.34) SLC6A2SLC6A4SLC6A3
SCHEMBL16026423 0.74 HTR3A (0.36) CYP2D6TSHRHTR1AADRA2ASLC6A2
SCHEMBL27432364 0.74 OPRM1 (0.34) OPRM1ADCY5
SCHEMBL11555527 0.74 CA2 (0.50) QDPRCYP3A4MEN1TSHRKMT2A
Piperazine SCHEMBL28078183 0.73 ADRB1 (0.37) CYP2D6TSHRHTR1AADRA2ASLC6A2
Hydrochloric Acid SCHEMBL27459404 0.73 HTR2C (0.36) OPRM1
Hydrochloric Acid SCHEMBL11553193 0.73 ESR2 (0.37) DRD1KDM4EDRD2RECQLMAPT
Hydrochloric Acid SCHEMBL11551113 0.73 TSHR (0.49) QDPRCYP3A4MEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4166180-A 2-ARYLPIPERAZINE DERIVATIVES AND THE PREPARATION THEREOF HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1979-08-28 US disclosed