SCHEMBL11567437

SCHEMBL11567437

COc1cc2c(cc1OC)C(C)(CCCN1CCN(c3ccccc3C)CC1)OCC2

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.49
DRD3 P35462 5/20 0.49
DRD4 P21917 3/20 0.49
HTR7 P34969 5/20 0.45
HTR2A P28223 5/20 0.45
HTR1A P08908 5/20 0.44
ADRA1A P35348 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9132075 0.85 DRD2 (0.48) DRD2DRD3DRD4HTR7HTR2A
SCHEMBL9130488 0.85 DRD2 (0.46) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL10752570 0.83 HTR1A (0.54) DRD2DRD3DRD4HTR7HTR2A
SCHEMBL9131769 0.83 DRD2 (0.44) DRD2DRD3DRD4HTR7HTR2A
SCHEMBL10749348 0.82 KDM4E (0.47) DRD2DRD3DRD4HTR7HTR2A
SCHEMBL9131510 0.81 DRD2 (0.45) DRD2DRD3DRD4HTR7HTR2A
SCHEMBL10744900 0.77 HTR7 (0.44) DRD3HTR7HTR1A
SCHEMBL10758269 0.76 DRD4 (0.47) DRD2DRD3DRD4HTR1AADRA1A
SCHEMBL11567096 0.75 ADORA2A (0.36) DRD2DRD3DRD4
SCHEMBL11674004 0.73 SIGMAR1 (0.42) DRD2DRD3DRD4HTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US claimed