SCHEMBL11575495

SCHEMBL11575495

CN1CCC(=C2c3ccccc3Sc3ccc(C#N)cc32)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SETD7 Q8WTS6 5/20 0.70
CHRM2 P08172 5/20 0.70
ADRA2A P08913 5/20 0.70
CHRM1 P11229 5/20 0.70
DRD1 P21728 5/20 0.70
ADRA1A P35348 5/20 0.70
DRD3 P35462 5/20 0.70
KCNH2 Q12809 5/20 0.70
HTR1A P08908 4/20 0.70
SLC6A2 P23975 4/20 0.70
SLC6A4 P31645 4/20 0.70
SLC6A3 Q01959 4/20 0.70
CYP2D6 P10635 3/20 0.70
CYP2C19 P33261 3/20 0.70
TBXA2R P21731 3/20 0.70
OPRM1 P35372 3/20 0.70
ADORA3 P0DMS8 1/20 0.70
HTT P42858 2/20 0.57
CYP3A4 P08684 2/20 0.57
DRD2 P14416 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL11574698 0.90 CYP3A4 (0.76) SETD7CHRM2ADRA2ACHRM1DRD1
Fumaric Acid SCHEMBL11574700 0.90 CYP3A4 (0.76) SETD7CHRM2ADRA2ACHRM1DRD1
Citatepine SCHEMBL2112235 0.85 DRD2 (0.51) SETD7CHRM2ADRA2ACHRM1DRD1
Pimethixene SCHEMBL29433731 0.84 SETD7 (1.00) SETD7CHRM2ADRA2ACHRM1DRD1
Pimethixene SCHEMBL301596 0.84 SETD7 (1.00) SETD7CHRM2ADRA2ACHRM1DRD1
SCHEMBL11432245 0.81 HTR1A (0.76) SETD7CHRM2ADRA2ACHRM1DRD1
SCHEMBL11574284 0.81 SETD7 (0.76) SETD7CHRM2ADRA2ACHRM1DRD1
SCHEMBL11520204 0.81 SETD7 (0.68) SETD7CHRM2ADRA2ACHRM1DRD1
SCHEMBL11575971 0.81 SETD7 (0.76) SETD7CHRM2ADRA2ACHRM1DRD1
SCHEMBL11431794 0.79 SETD7 (0.72) SETD7CHRM2ADRA2ACHRM1DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4086350-A FLUORO, CHLORO AND CYANO SUBSTITUTED 4-(9-XANTHENYLIDENE, 9-THIOXANTHENYLIDENE OR 11(6H)-DIBENZO(B,E)OXEPINYLIDENE)-1-METHYL-PIPERIDINES SMITHKLINE CORPORATION (US) 1978-04-25 US claimed
US-4086350-A FLUORO, CHLORO AND CYANO SUBSTITUTED 4-(9-XANTHENYLIDENE, 9-THIOXANTHENYLIDENE OR 11(6H)-DIBENZO(B,E)OXEPINYLIDENE)-1-METHYL-PIPERIDINES SMITHKLINE CORPORATION (US) 1978-04-25 US disclosed
US-4076714-A 1-Methyl-4-(2-carboxy-thioxanthen-9-ylidene)-piperidine an appetite stimulant and antihistaminic agent MERCK & CO., INC. (US) 1978-02-28 US disclosed