SCHEMBL11620971

SCHEMBL11620971

C1=C(CCCN2CCCC2)c2ccccc2C1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.54
GRIN2B Q13224 2/20 0.47
LTA4H P09960 1/20 0.46
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SLC6A3 Q01959 1/20 0.42
HTR6 P50406 1/20 0.42
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11542289 0.98 SIGMAR1 (0.53) SIGMAR1GRIN2BLTA4HALDH1A1L3MBTL1
SCHEMBL13297902 0.92 SLC6A3 (0.50) SIGMAR1SLC6A3HTR6
SCHEMBL11542316 0.90 SIGMAR1 (0.51) SIGMAR1SLC6A3HTR6
SCHEMBL9304524 0.87 SIGMAR1 (0.55) SIGMAR1HTR6
SCHEMBL3868123 0.81 HTR6 (0.53) SIGMAR1ALDH1A1HTR6
SCHEMBL3874874 0.81 HTR6 (0.53) SIGMAR1ALDH1A1HTR6
SCHEMBL11541639 0.80 SIGMAR1 (0.48) SIGMAR1GRIN2B
SCHEMBL9304462 0.78 CNR1 (0.50) SIGMAR1
SCHEMBL31121639 0.77 HTR6 (0.56) SIGMAR1HTR6
SCHEMBL2338975 0.77 HTR6 (0.56) SIGMAR1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4127578-A Diene intermediates for indantetrols E. R. SQUIBB & SONS, INC. (US) 1978-11-28 US disclosed
US-4092318-A HYPOTENSIVES E. R. SQUIBB & SONS, INC. (US) 1978-05-30 US disclosed
US-4044040-A HYPERTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1977-08-23 US disclosed