SCHEMBL11713243

SCHEMBL11713243

Nc1nc2cc(-c3c(Cl)cccc3Cl)ccc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 5/20 0.50
CACNG8 Q8WXS5 5/20 0.50
NUDT1 P36639 3/20 0.47
MASP2 O00187 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
AOC3 Q16853 1/20 0.47
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
HTR3A P46098 1/20 0.46
BACE1 P56817 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
SRC P12931 2/20 0.46
FABP6 P51161 1/20 0.41
PTPN11 Q06124 1/20 0.41
TYMS P04818 1/20 0.40
ABL1 P00519 1/20 0.40
PLAU P00749 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11713250 0.88 HTR3E (0.58) GRIA1CACNG8NUDT1MASP2MEN1
SCHEMBL5678732 0.83 JAK2 (0.55) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL117352 0.81 BACE1 (0.54) NUDT1MASP2MEN1ALDH1A1KMT2A
Bromide SCHEMBL2381776 0.80 BACE1 (0.53) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL5679783 0.79 BACE1 (0.59) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL14655239 0.77 HTR3E (0.49) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL3827667 0.77 ALDH1A1 (0.58) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL5680955 0.75 XDH (0.52) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL5681861 0.75 ALDH1A1 (0.47) NUDT1MASP2MEN1ALDH1A1KMT2A
SCHEMBL5679180 0.75 TAAR1 (0.50) NUDT1MASP2MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4004016-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1977-01-18 US disclosed
US-3981886-A Amino-benzimidazole derivatives E. R. SQUIBB & SONS, INC. (US) 1976-09-21 US disclosed