SCHEMBL1191749

SCHEMBL1191749

CC1(C)C(=O)N(c2ccc(C#N)cc2)C(=O)N1Cc1ccccc1Oc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.45
TAS2R8 Q9NYW2 5/20 0.44
ELANE P08246 1/20 0.43
MCHR1 Q99705 1/20 0.41
PGR P06401 2/20 0.40
IGF1R P08069 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
POLB P06746 1/20 0.38
FAAH O00519 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021401 0.89 TAS2R8 (0.46) SLC6A4TAS2R8IGF1RFAAH
SCHEMBL8023307 0.89 TAS2R8 (0.47) SLC6A4TAS2R8ELANEIGF1RFAAH
SCHEMBL12873209 0.89 MCHR1 (0.45) SLC6A4TAS2R8MCHR1
SCHEMBL12873200 0.88 TAS2R8 (0.41) TAS2R8IGF1RFAAH
SCHEMBL8023309 0.87 TAS2R8 (0.46) SLC6A4TAS2R8ELANEIGF1RFAAH
SCHEMBL8019464 0.87 TAS2R8 (0.44) SLC6A4TAS2R8MCHR1IGF1RFAAH
SCHEMBL8010593 0.87 TAS2R8 (0.44) SLC6A4TAS2R8IGF1RFAAH
SCHEMBL8001620 0.86 LMNA (0.46) SLC6A4TAS2R8IGF1RFAAH
SCHEMBL8027028 0.86 HTR2A (0.47) SLC6A4TAS2R8ELANEIGF1RFAAH
SCHEMBL12873224 0.86 TAS2R8 (0.48) SLC6A4TAS2R8ELANEPGRIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-02-24 US disclosed
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-02-24 US disclosed
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-02-24 US disclosed
EP-2252592-A1 ARYLCHALCOGENO-ARYLALKYL-SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF Sanofi-Aventis (FR) 2010-11-24 EP disclosed
WO-2009097998-A1 ARYLCHALCOGENO-ARYLALKYL-SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof PGC, LIPC, CEL SLC6A4 3548/4885TAS2R8 318/4885ELANE 754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.